SCHEMBL7092945

SCHEMBL7092945

Nc1nc(Nc2ccc(C(=O)Cl)cc2)nn1C(=O)c1ccccc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNB2 O95067 3/20 0.71
CDK1 P06493 3/20 0.71
CCNB1 P14635 3/20 0.71
CCNB3 Q8WWL7 3/20 0.71
JAK1 P23458 7/20 0.61
TYK2 P29597 7/20 0.61
JAK2 O60674 7/20 0.61
JAK3 P52333 5/20 0.61
F12 P00748 2/20 0.50
F2 P00734 1/20 0.50
PLK4 O00444 1/20 0.50
STK25 O00506 1/20 0.50
RIOK3 O14730 1/20 0.50
AURKA O14965 1/20 0.50
GAK O14976 1/20 0.50
DCLK1 O15075 1/20 0.50
PDPK1 O15530 1/20 0.50
DAPK3 O43293 1/20 0.50
NUAK1 O60285 1/20 0.50
ROCK2 O75116 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1248143 0.90 CCNB2 (0.77) CCNB2CDK1CCNB1CCNB3JAK1
SCHEMBL1248356 0.86 CCNB2 (0.65) CCNB2CDK1CCNB1CCNB3JAK1
SCHEMBL1250806 0.85 CCNB2 (0.67) CCNB2CDK1CCNB1CCNB3JAK1
SCHEMBL1167320 0.84 CCNB2 (0.62) CCNB2CDK1CCNB1CCNB3JAK1
SCHEMBL1167929 0.84 CCNB2 (0.65) CCNB2CDK1CCNB1CCNB3JAK1
SCHEMBL1249224 0.84 CCNB2 (0.65) CCNB2CDK1CCNB1CCNB3JAK1
SCHEMBL5726202 0.83 CCNB2 (1.00) CCNB2CDK1CCNB1CCNB3JAK1
SCHEMBL1167961 0.82 CCNB2 (0.62) CCNB2CDK1CCNB1CCNB3JAK1
SCHEMBL5964782 0.81 TYK2 (0.62) CCNB2CDK1CCNB1CCNB3JAK1
SCHEMBL1248362 0.81 TYK2 (0.63) CCNB2CDK1CCNB1CCNB3JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1355889-A1 SUBSTITUTED TRIAZOLE DIAMINE DERIVATIVES AS KINASE INHIBITORS Ortho-McNeil Pharmaceutical, Inc. (US) 2003-10-29 EP disclosed
WO-2002057240-A1 SUBSTITUTED TRIAZOLE DIAMINE DERIVATIVES AS KINASE INHIBITORS ORTHO MC NEIL PHARMACEUTICAL, INC. (US) 2002-07-25 WO disclosed