SCHEMBL7093701

SCHEMBL7093701

CC(C)c1ccc(Cc2c(N)nc(SCCN3CCNCC3)nc2N)cc1

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 14/20 0.53
HTR2C P28335 14/20 0.53
ALOX15 P16050 1/20 0.38
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HTR6 P50406 1/20 0.36
HTR1D P28221 1/20 0.36
HTR1B P28222 1/20 0.36
SLC6A4 P31645 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Water SCHEMBL7092927 0.84 HTR2A (0.71) HTR2AHTR2CALDH1A1HTR6
Hydrochloric Acid SCHEMBL7096035 0.83 HTR2A (0.52) HTR2AHTR2CALOX15SLC6A4
Hydrochloric Acid SCHEMBL7093198 0.80 HRH3 (0.50) HTR2AHTR2CKDM4EALDH1A1
Hydrochloric Acid SCHEMBL7096651 0.77 HTR2A (0.46) HTR2AHTR2CSLC6A4
Hydrochloric Acid SCHEMBL7096922 0.77 HTR2A (0.46) HTR2AHTR2CKDM4EALDH1A1
Hydrochloric Acid SCHEMBL7097609 0.77 HTR2A (0.62) HTR2AHTR2CALDH1A1
SCHEMBL7096779 0.75 HTR2A (0.71) HTR2AHTR2CALOX15KDM4EALDH1A1
SCHEMBL7099072 0.74 HTR2A (0.69) HTR2AHTR2CHTR6
Hydrochloric Acid SCHEMBL7591093 0.70 HTR2A (0.59) HTR2AHTR2C
Hydrochloric Acid SCHEMBL7097961 0.70 HTR2A (0.54) HTR2AHTR2CSLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1194415-B1 NOVEL PIPERAZINYLALKYLTHIOPYRIMIDINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME, AND A PROCESS FOR THEIR PREPARATION EGYT GYOGYSZERVEGYESZETI GYAR (HU) 2003-08-20 EP disclosed
US-6469168-B1 FOR THE TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS, ESPECIALLY ANXIETY EGIS Gyógyszergyár Rt. (HU) 2002-10-22 US disclosed