SCHEMBL7096091

SCHEMBL7096091

O=C1N[C@@H](O)[C@@H](O)N1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10746362 1.00
SCHEMBL30007 1.00
SCHEMBL10746346 1.00
SCHEMBL9736596 0.83 CRBN (0.33)
SCHEMBL22733469 0.80 IDUA (0.31)
SCHEMBL21229510 0.78
SCHEMBL5081619 0.74
SCHEMBL48373 0.70 TSHR (0.44)
SCHEMBL16253387 0.69
SCHEMBL36249 0.67 MAPT (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923560-B1 BRIDGED AND POSSIBLY METHYLOLIZED 4,5-BIS-DI-HIDROXY-IMIDAZOLIDIN-2-ONES, PROCESS FOR THEIR PRODUCTION AND USE THEREOF BASF AG (DE) 2003-01-08 EP claimed
US-6153762-A IMPROVE CREASE RECOVERY, WRICKLE RESISTANCE AND REDUCE TEXTILE SHRINKAGE, IMPROVE THE STRENGTH OF THE FABRIC, REDUCING THE USE OF FORMALDEHYDE BASF AKTIENGESELLSCHAFT (DE) 2000-11-28 US claimed
EP-0923560-A1 BRIDGED AND POSSIBLY METHYLOLIZED 4,5-BIS-DI-HIDROXY-IMIDAZOLIDIN-2-ONES, PROCESS FOR THEIR PRODUCTION AND USE THEREOF BASF AKTIENGESELLSCHAFT (DE) 1999-06-23 EP claimed
WO-1998005650-A1 BRIDGED AND POSSIBLY METHYLOLIZED 4,5-BIS-DI-HYDROXY-IMIDAZOLIDIN-2-ONES, PROCESS FOR THEIR PRODUCTION AND USE THEREOF BASF AKTIENGESELLSCHAFT (DE) 1998-02-12 WO claimed
US-9944769-B2 Urea-derived products and methods for making same THE PROCTER & GAMBLE COMPANY (US) 2018-04-17 US disclosed
US-9944769-B2 Urea-derived products and methods for making same THE PROCTER & GAMBLE COMPANY (US) 2018-04-17 US disclosed
EP-2920152-B1 UREA-DERIVED PRODUCTS AND METHODS FOR MAKING SAME PROCTER & GAMBLE (US) 2016-06-29 EP disclosed
US-20140117274-A1 UREA-DERIVED PRODUCTS AND METHODS FOR MAKING SAME THE PROCTER & GAMBLE COMPANY (US) 2014-05-01 US disclosed
US-20140117274-A1 UREA-DERIVED PRODUCTS AND METHODS FOR MAKING SAME THE PROCTER & GAMBLE COMPANY (US) 2014-05-01 US disclosed
WO-2014066583-A1 UREA-DERIVED PRODUCTS AND METHODS FOR MAKING SAME THE PROCTER & GAMBLE COMPANY (US) 2014-05-01 WO disclosed
EP-0923560-B1 BRIDGED AND POSSIBLY METHYLOLIZED 4,5-BIS-DI-HIDROXY-IMIDAZOLIDIN-2-ONES, PROCESS FOR THEIR PRODUCTION AND USE THEREOF BASF AG (DE) 2003-01-08 EP disclosed
EP-0923560-B1 BRIDGED AND POSSIBLY METHYLOLIZED 4,5-BIS-DI-HIDROXY-IMIDAZOLIDIN-2-ONES, PROCESS FOR THEIR PRODUCTION AND USE THEREOF BASF AG (DE) 2003-01-08 EP disclosed
US-6153762-A IMPROVE CREASE RECOVERY, WRICKLE RESISTANCE AND REDUCE TEXTILE SHRINKAGE, IMPROVE THE STRENGTH OF THE FABRIC, REDUCING THE USE OF FORMALDEHYDE BASF AKTIENGESELLSCHAFT (DE) 2000-11-28 US disclosed
US-6153762-A IMPROVE CREASE RECOVERY, WRICKLE RESISTANCE AND REDUCE TEXTILE SHRINKAGE, IMPROVE THE STRENGTH OF THE FABRIC, REDUCING THE USE OF FORMALDEHYDE BASF AKTIENGESELLSCHAFT (DE) 2000-11-28 US disclosed
EP-0923560-A1 BRIDGED AND POSSIBLY METHYLOLIZED 4,5-BIS-DI-HIDROXY-IMIDAZOLIDIN-2-ONES, PROCESS FOR THEIR PRODUCTION AND USE THEREOF BASF AKTIENGESELLSCHAFT (DE) 1999-06-23 EP disclosed
EP-0923560-A1 BRIDGED AND POSSIBLY METHYLOLIZED 4,5-BIS-DI-HIDROXY-IMIDAZOLIDIN-2-ONES, PROCESS FOR THEIR PRODUCTION AND USE THEREOF BASF AKTIENGESELLSCHAFT (DE) 1999-06-23 EP disclosed
WO-1998005650-A1 BRIDGED AND POSSIBLY METHYLOLIZED 4,5-BIS-DI-HYDROXY-IMIDAZOLIDIN-2-ONES, PROCESS FOR THEIR PRODUCTION AND USE THEREOF BASF AKTIENGESELLSCHAFT (DE) 1998-02-12 WO disclosed
WO-1998005650-A1 BRIDGED AND POSSIBLY METHYLOLIZED 4,5-BIS-DI-HYDROXY-IMIDAZOLIDIN-2-ONES, PROCESS FOR THEIR PRODUCTION AND USE THEREOF BASF AKTIENGESELLSCHAFT (DE) 1998-02-12 WO disclosed
US-4421546-A HERBICIDES FOR AQUATIC VEGETATION ELI LILLY AND COMPANY (US) 1983-12-20 US disclosed
US-4354030-A CONTROL OF AQUATIC VEGETATION ELI LILLY AND COMPANY (US) 1982-10-12 US disclosed