SCHEMBL7096517

SCHEMBL7096517

Nc1nc(-c2ccco2)c2cnn(Cc3ccsc3S(=O)(=O)Nc3ccccc3)c2n1

nearest known ligand 0.60

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 20/20 0.60
ADORA1 P30542 18/20 0.60
HDAC1 Q13547 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4557673 0.79 ADORA2A (0.64) ADORA2AADORA1HDAC1
SCHEMBL4452012 0.76 ADORA2A (1.00) ADORA2AADORA1HDAC1
SCHEMBL4452013 0.76 ADORA2A (1.00) ADORA2AADORA1HDAC1
SCHEMBL4450557 0.74 ADORA2A (1.00) ADORA2AADORA1
SCHEMBL4452784 0.74 ADORA2A (1.00) ADORA2AADORA1HDAC1
SCHEMBL13601276 0.73 ADORA2A (0.60) ADORA2AADORA1HDAC1
SCHEMBL4458505 0.73 ADORA2A (0.64) ADORA2AADORA1HDAC1
SCHEMBL4459531 0.73 ADORA2A (1.00) ADORA2AADORA1
SCHEMBL4459074 0.72 ADORA2A (1.00) ADORA2AADORA1HDAC1
SCHEMBL4464120 0.72 ADORA2A (0.61) ADORA2AADORA1HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1349552-A1 PYRAZOLO 3,4-D]PYRIMIDINE DERIVATIVES AND THEIR USE AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2003-10-08 EP disclosed
WO-2002055082-A1 PYRAZOLO[3,4-D]PYRIMIDINE DERIVATIVES AND THEIR USE AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2002-07-18 WO disclosed