SCHEMBL7102594

SCHEMBL7102594

COc1ccc(COc2[c]c(F)ccc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAOB P27338 5/20 0.49
APP P05067 8/20 0.47
NPC1 O15118 3/20 0.44
RAB9A P51151 3/20 0.44
TDP1 Q9NUW8 1/20 0.44
IDO1 P14902 2/20 0.43
AGXT P21549 2/20 0.43
HTR1A P08908 1/20 0.43
ADRA1D P25100 1/20 0.43
ADRA1A P35348 1/20 0.43
ADRA1B P35368 1/20 0.43
POLB P06746 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28550433 0.85 MAOB (0.53) MAOBAPPNPC1RAB9ATDP1
SCHEMBL17260899 0.82 MAPT (0.43) MAOBRAB9ATDP1HTR1ASMN1; SMN2
SCHEMBL7024020 0.81 MAOB (0.53) MAOBAPPNPC1RAB9ATDP1
SCHEMBL5568926 0.77 TDP1 (0.44) MAOBAPPNPC1RAB9ATDP1
SCHEMBL7015864 0.76 TLR4 (0.48) MAOBAPPNPC1RAB9ATDP1
SCHEMBL2451926 0.74 APP (0.49) MAOBAPPNPC1RAB9ATDP1
SCHEMBL160707 0.73
SCHEMBL21680729 0.73 PTPN1 (0.38) SMN1; SMN2
SCHEMBL159421 0.72 NQO1 (0.36) TDP1SMN1; SMN2
SCHEMBL6195407 0.71 MAOB (0.51) MAOBTDP1HTR1AADRA1DADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1326856-A1 PYRIDINE DERIVATIVES WITH IKB-KINASE (IKK-BETA) INHIBITING ACTIVITY Bayer Aktiengesellschaft (DE) 2003-07-16 EP disclosed
WO-2002024679-A1 PYRIDINE DERIVATIVES WITH IKB-KINASE (IKK-β) INHIBITING ACTIVITY BAYER AKTIENGESELLSCHAFT (DE) 2002-03-28 WO disclosed