SCHEMBL7103997

SCHEMBL7103997

CC(C)(C)OC(=O)C1(C)CCC(C(=O)N[C@@H](Cc2ccc(NC(=O)c3c(Cl)cccc3Cl)cc2)C(=O)O)C1(C)C

nearest known ligand 0.55

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 20/20 0.55
ITGA4 P13612 20/20 0.55
ITGA2 P17301 1/20 0.53
ITGB7 P26010 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7104001 1.00 ITGB1 (0.55) ITGB1ITGA4ITGA2ITGB7
SCHEMBL7098743 0.94 ITGB1 (0.49) ITGB1ITGA4ITGA2ITGB7
SCHEMBL7098745 0.94 ITGB1 (0.49) ITGB1ITGA4ITGA2ITGB7
SCHEMBL7247044 0.94 ITGB1 (0.49) ITGB1ITGA4ITGA2ITGB7
SCHEMBL7247043 0.94 ITGB1 (0.49) ITGB1ITGA4ITGA2ITGB7
SCHEMBL7098677 0.89 ITGB1 (0.59) ITGB1ITGA4ITGA2ITGB7
SCHEMBL7098060 0.89 ITGB1 (0.59) ITGB1ITGA4ITGA2ITGB7
SCHEMBL7100655 0.89 ITGB1 (0.59) ITGB1ITGA4ITGA2ITGB7
SCHEMBL7097651 0.89 ITGB1 (0.59) ITGB1ITGA4ITGA2ITGB7
SCHEMBL7104171 0.89 ITGB1 (0.59) ITGB1ITGA4ITGA2ITGB7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991619-B1 INHIBITORS OF ALPHA 4-BETA 1 MEDIATED CELL ADHESION TANABE SEIYAKU CO (JP) 2003-09-10 EP disclosed
US-6596752-B1 Small molecules that are potent inhibitors of alpha 4 beta 1 mediated adhesion to either VCAM or CS-1 and which could be useful for the treatment of inflammatory diseases. TANABE SEIYAKU CO., LTD. (JP) 2003-07-22 US disclosed
US-6482849-B1 Inhibitors of α4β1 mediated cell adhesion TANABE SEIYAKU CO., LTD. (JP) 2002-11-19 US disclosed