SCHEMBL7104760

SCHEMBL7104760

CCCCCC/C=C(/OC)O[Si](C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EP300 Q09472 1/20 0.40
TSHR P16473 2/20 0.34
EPHX1 P07099 1/20 0.32
POLB P06746 2/20 0.32
LPAR1 Q92633 1/20 0.32
LPAR2 Q9HBW0 1/20 0.32
LPAR3 Q9UBY5 1/20 0.32
POLA1 P09884 1/20 0.32
TERT O14746 2/20 0.32
GMNN O75496 1/20 0.32
USP2 O75604 1/20 0.32
LMNA P02545 1/20 0.32
CYP1A2 P05177 1/20 0.32
MAPT P10636 1/20 0.32
CYP2C9 P11712 1/20 0.32
ALOX15 P16050 1/20 0.32
APEX1 P27695 1/20 0.32
CYP2C19 P33261 1/20 0.32
RECQL P46063 1/20 0.32
BLM P54132 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7104762 1.00 EP300 (0.40) EP300TSHREPHX1POLBLPAR1
SCHEMBL16295144 0.90 EP300 (0.44) EP300TSHRPOLBTERTGMNN
SCHEMBL3589901 0.84
SCHEMBL9913422 0.84
SCHEMBL9718334 0.84 EP300 (0.48) EP300TSHREPHX1POLBTERT
SCHEMBL4583581 0.84 EP300 (0.48) EP300TSHREPHX1POLBTERT
SCHEMBL14721325 0.81 EP300 (0.37) EP300TSHRPOLBGMNNUSP2
SCHEMBL16782695 0.81 EP300 (0.37) EP300TSHRPOLBGMNNUSP2
SCHEMBL14721323 0.81 EP300 (0.37) EP300TSHRPOLBGMNNUSP2
SCHEMBL3933343 0.79 EP300 (0.44) EP300TSHREPHX1POLBTERT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1127886-B1 Synthesis of 3,6-dialkyl-5,6-dihydro-4-hydroxy-2H-pyran-2one HOFFMANN LA ROCHE (CH) 2003-05-07 EP disclosed
US-6552204-B1 Lactonization of an acyl halide and a ketene acetal or reacting acyl halide with malonate half acid then cyclizing; high yield ROCHE COLORADO CORPORATION 2003-04-22 US disclosed
CN-1319596-A Synthesis of 3,6-dialkyl 5,6-dihydro-4-hydroxide-2H-pyran-2-ketone HOFFMANN LA ROCHE (CH) 2001-10-31 CN disclosed
EP-1127886-A1 Synthesis of 3,6-dialkyl-5,6-dihydro-4-hydroxy-2H-pyran-2one F. HOFFMANN-LA ROCHE AG (CH) 2001-08-29 EP disclosed