SCHEMBL7108371

SCHEMBL7108371

Oc1cccc(-c2sc3cc(O)ccc3c2Oc2ccc(OCCN3CCCCC3)cc2)c1

nearest known ligand 0.87

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 20/20 0.87
ESR2 Q92731 19/20 0.87
MEN1 O00255 1/20 0.61
PLD2 O14939 1/20 0.61
KDM1A O60341 1/20 0.61
NR1I2 O75469 1/20 0.61
USP2 O75604 1/20 0.61
ALDH1A1 P00352 1/20 0.61
C5 P01031 1/20 0.61
LMNA P02545 1/20 0.61
TP53 P04637 1/20 0.61
FYN P06241 1/20 0.61
PGR P06401 1/20 0.61
CYP3A4 P08684 1/20 0.61
ADRA2A P08913 1/20 0.61
ADORA3 P0DMS8 1/20 0.61
CYP2D6 P10635 1/20 0.61
MAPT P10636 1/20 0.61
CYP2C9 P11712 1/20 0.61
ADRB3 P13945 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7103336 0.99 ESR1 (0.86) ESR1ESR2MEN1PLD2KDM1A
Hydrochloric Acid SCHEMBL7106595 0.98 ESR1 (0.84) ESR1ESR2MEN1ALDH1A1LMNA
SCHEMBL6552026 0.93 ESR1 (1.00) ESR1ESR2MEN1PLD2KDM1A
SCHEMBL7108651 0.93 ESR1 (0.79) ESR1ESR2
SCHEMBL7103407 0.92 ESR1 (0.78) ESR1ESR2
Hydrochloric Acid SCHEMBL7976502 0.92 ESR1 (0.98) ESR1ESR2MEN1PLD2KDM1A
SCHEMBL7106179 0.92 ESR1 (0.83) ESR1ESR2
Hydrochloric Acid SCHEMBL7107405 0.92 ESR1 (0.77) ESR1ESR2
Hydrochloric Acid SCHEMBL7100898 0.91 ESR1 (0.76) ESR1ESR2
SCHEMBL3743164 0.91 ESR1 (1.00) ESR1ESR2MEN1PLD2KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0827959-B1 Benzo[B]thiophene compounds, intermediates, processes, compositions, and methods LILLY CO ELI (US) 2003-12-03 EP disclosed
US-5977382-A Benzo[b]thiophene compounds, intermediates, processes, compositions, and methods ELI LILLY AND COMPANY (US) 1999-11-02 US disclosed
US-5977098-A Benzo[B]thiophene compounds, intermediates, processes, compositions, and methods ELI LILLY AND COMPANY (US) 1999-11-02 US disclosed
EP-0827959-A2 Benzo[B]thiophene compounds, intermediates, processes, compositions, and methods ELI LILLY AND COMPANY (US) 1998-03-11 EP disclosed