SCHEMBL7111397

SCHEMBL7111397

CC/C(=C(/c1ccc(I)cc1)c1ccc(OCCN2C=C2)cc1)c1ccccc1

nearest known ligand 0.73

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PDE1A P54750 16/20 0.73
PDE1B Q01064 16/20 0.73
PDE1C Q14123 16/20 0.73
ESR1 P03372 1/20 0.73
ESR2 Q92731 1/20 0.73
CYP3A4 P08684 1/20 0.64
CYP19A1 P11511 1/20 0.64
PSMB1 P20618 2/20 0.63
PSMB5 P28074 1/20 0.63
PSMB2 P49721 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7148860 1.00 PDE1A (0.73) PDE1APDE1BPDE1CESR1ESR2
SCHEMBL407938 0.87 PDE1A (0.72) PDE1APDE1BPDE1CESR1ESR2
SCHEMBL285263 0.87 PDE1A (0.72) PDE1APDE1BPDE1CESR1ESR2
SCHEMBL285264 0.87 PDE1A (0.72) PDE1APDE1BPDE1CESR1ESR2
SCHEMBL18291033 0.86 CYP19A1 (0.87) PDE1APDE1BPDE1CESR1ESR2
Idoxifene SCHEMBL19217 0.85 PDE1A (1.00) PDE1APDE1BPDE1CESR1ESR2
Idoxifene SCHEMBL19216 0.85 PDE1A (1.00) PDE1APDE1BPDE1CESR1ESR2
Idoxifene SCHEMBL3774574 0.85 PDE1A (1.00) PDE1APDE1BPDE1CESR1ESR2
SCHEMBL10349389 0.84 PDE1A (0.73) PDE1APDE1BPDE1CESR1ESR2
SCHEMBL10608838 0.84 PDE1A (0.73) PDE1APDE1BPDE1CESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1023264-B1 NEW MARKER, PRODUCTION PROCESS AND USE THEREOF QUIVY JACQUES (BE) 2003-03-19 EP claimed
EP-1023264-B1 NEW MARKER, PRODUCTION PROCESS AND USE THEREOF QUIVY JACQUES (BE) 2003-03-19 EP disclosed