Terpyridine

Terpyridine

SCHEMBL7112915

[Pt].c1ccc(-c2cccc(-c3ccccn3)n2)nc1.c1ccc(-c2cccc(-c3ccccn3)n2)nc1

nearest known ligand 0.95

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 9/20 0.95
TP53 P04637 4/20 0.95
ALOX15 P16050 4/20 0.95
L3MBTL1 Q9Y468 4/20 0.95
SMN1; SMN2 Q16637 4/20 0.95
CCR1 P32246 3/20 0.95
CCR5 P51681 3/20 0.95
CCR8 P51685 3/20 0.95
LMNA P02545 3/20 0.95
TDP1 Q9NUW8 3/20 0.95
HTT P42858 2/20 0.95
ALPL P05186 2/20 0.95
HSP90AA1 P07900 1/20 0.95
ALPI P09923 1/20 0.95
ALPG P10696 1/20 0.95
MAPK1 P28482 1/20 0.95
CYP1A2 P05177 2/20 0.74
POLB P06746 1/20 0.74
METAP1 P53582 1/20 0.74
BLM P54132 1/20 0.74

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Terpyridine SCHEMBL1616654 1.00 KDM4E (0.95) KDM4ETP53ALOX15L3MBTL1SMN1; SMN2
SCHEMBL30172832 0.97 KDM4E (1.00) KDM4ETP53ALOX15L3MBTL1SMN1; SMN2
Terpyridine SCHEMBL57442 0.97 KDM4E (1.00) KDM4ETP53ALOX15L3MBTL1SMN1; SMN2
SCHEMBL7964803 0.97 KDM4E (1.00) KDM4ETP53ALOX15L3MBTL1SMN1; SMN2
Terpyridine SCHEMBL29357603 0.97 KDM4E (1.00) KDM4ETP53ALOX15L3MBTL1SMN1; SMN2
Terpyridine SCHEMBL3150051 0.95 KDM4E (0.95) KDM4ETP53ALOX15L3MBTL1SMN1; SMN2
Terpyridine SCHEMBL8536195 0.95 KDM4E (0.95) KDM4ETP53ALOX15L3MBTL1SMN1; SMN2
Terpyridine SCHEMBL31621745 0.95 KDM4E (0.95) KDM4ETP53ALOX15L3MBTL1SMN1; SMN2
Terpyridine SCHEMBL2953496 0.95 KDM4E (0.95) KDM4ETP53ALOX15L3MBTL1SMN1; SMN2
Terpyridine SCHEMBL5899140 0.95 KDM4E (0.95) KDM4ETP53ALOX15L3MBTL1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1144423-B1 BIS-TERPYRIDINE-PLATINUM(II) COMPLEXES ISIS INNOVATION (GB) 2003-10-22 EP disclosed
EP-1144423-A1 BIS-TERPYRIDINE-PLATINUM(II) COMPLEXES ISIS INNOVATION LIMITED (GB) 2001-10-17 EP disclosed
WO-2000043405-A1 BIS-TERPYRIDINE-PLATINUM(II) COMPLEXES ISIS INNOVATION LIMITED (GB) 2000-07-27 WO disclosed