SCHEMBL7116226

SCHEMBL7116226

CS(=O)(=O)N1CCN(Cc2cccc3[nH]c(-n4c(=O)ccc5ccccc54)cc23)CC1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.43
GPR84 Q9NQS5 1/20 0.41
HTR6 P50406 9/20 0.40
KDM4E B2RXH2 4/20 0.39
ALOX15 P16050 1/20 0.39
HTT P42858 1/20 0.39
CYP2D6 P10635 3/20 0.38
CYP3A4 P08684 2/20 0.38
TSHR P16473 1/20 0.38
LMNA P02545 1/20 0.38
OPRM1 P35372 1/20 0.36
OPRK1 P41145 1/20 0.36
PTGER3 P43115 1/20 0.36
ALDH1A1 P00352 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
AKT1 P31749 1/20 0.36
ESR1 P03372 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14311030 0.77 NPSR1 (0.50) NPSR1KDM4EALOX15HTTCYP2D6
SCHEMBL149448 0.76 KDR (0.51) NPSR1GPR84KDM4EALOX15HTT
SCHEMBL14286538 0.74 NPSR1 (0.47) NPSR1HTR6KDM4EALOX15HTT
SCHEMBL144879 0.66 CHEK1 (0.50) NPSR1HTR6OPRM1OPRK1
SCHEMBL143698 0.66 NPSR1 (0.43) NPSR1GPR84KDM4EALOX15HTT
SCHEMBL5058960 0.64 CHEK1 (0.52) NPSR1
SCHEMBL7116590 0.62 CHEK1 (0.46) KDM4ETSHRLMNAALDH1A1
SCHEMBL172902 0.61 CHEK1 (0.67)
SCHEMBL1029651 0.60 RECQL (0.73) KDM4ECYP2D6TSHRLMNAALDH1A1
Hydrochloric Acid SCHEMBL5677881 0.60 CHEK1 (0.66)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003020276-A1 TYROSINE KINASE INHIBITORS MERCK & CO., INC. (US) 2003-03-13 WO disclosed