SCHEMBL7118259

SCHEMBL7118259

O=C1CC(SSC2CC(=O)NC2=O)C(=O)N1

nearest known ligand 0.48

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAP3K14 Q99558 1/20 0.48
CRBN Q96SW2 17/20 0.40
SMN1; SMN2 Q16637 1/20 0.39
DDB1 Q16531 16/20 0.37
CYP19A1 P11511 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3800179 0.90 MAP3K14 (0.44) MAP3K14CRBNSMN1; SMN2DDB1CYP19A1
SCHEMBL22192782 0.86 MAP3K14 (0.41) MAP3K14CRBNSMN1; SMN2DDB1CYP19A1
Propionic Acid SCHEMBL2689345 0.82 SMN1; SMN2 (0.40) MAP3K14CRBNSMN1; SMN2DDB1
SCHEMBL13673930 0.82
SCHEMBL211974 0.80
SCHEMBL21305366 0.80
SCHEMBL1024468 0.80
SCHEMBL807677 0.80
SCHEMBL4774020 0.80
SCHEMBL22702164 0.75 MAP3K14 (0.40) MAP3K14CRBNSMN1; SMN2DDB1CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023157822-A1 RADIOACTIVE COMPLEX OF ANTI-VEGF ANTIBODY, AND RADIOPHARMACEUTICAL 日本メジフィジックス株式会社 2023-08-24 WO disclosed
WO-2023033022-A1 RADIOACTIVE COMPLEX OF DEGLYCOSYLATED ANTIBODY AND RADIOACTIVE PHARMACEUTICAL PRODUCT 日本メジフィジックス株式会社 2023-03-09 WO disclosed
WO-2023277144-A1 HUMANIZED ANTIBODY CAPABLE OF BINDING TO HEG1 PROTEIN, AND COMPLEX OF SAID ANTIBODY AND RADIOACTIVE NUCLEAR SPECIES 日本メジフィジックス株式会社 2023-01-05 WO disclosed
WO-2022224980-A1 RADIOACTIVE COMPLEX OF ANTI-CD20 ANTIBODY, AND RADIOPHARMACEUTICAL 日本メジフィジックス株式会社 2022-10-27 WO disclosed
WO-2022211051-A1 RADIOACTIVE COMPLEX OF ANTI-EGFR ANTIBODY, AND RADIOPHARMACEUTICAL 日本メジフィジックス株式会社 2022-10-06 WO disclosed
US-20030180957-A1 Target and method SENSE PROTEOMIC LIMITED 2003-09-25 US disclosed
WO-2003056344-A2 PROTEIN ANALYSIS USING MASS SPECTROMETRY SENSE PROTEOMIC LIMITED (GB) 2003-07-10 WO disclosed