SCHEMBL7128545

SCHEMBL7128545

CC[C@H](C(=O)N1C(=O)OC[C@@H]1Cc1ccccc1)[C@@H](C)CC

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 3/20 0.47
IL6ST P40189 1/20 0.43
FAAH O00519 1/20 0.41
ACE P12821 2/20 0.41
NAAA Q02083 1/20 0.41
IDH1 O75874 8/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
PPARG P37231 1/20 0.37
CSNK2B P67870 1/20 0.36
CSNK2A1 P68400 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29766885 0.92 PPARA (0.48) PPARAIL6STFAAHNAAAIDH1
SCHEMBL22686526 0.92 PPARA (0.48) PPARAIL6STFAAHNAAAIDH1
SCHEMBL22686525 0.92 PPARA (0.48) PPARAIL6STFAAHNAAAIDH1
SCHEMBL22686527 0.92 PPARA (0.48) PPARAIL6STFAAHNAAAIDH1
SCHEMBL26181174 0.91 PPARA (0.47) PPARAIL6STFAAHACENAAA
SCHEMBL27101415 0.91 PPARA (0.47) PPARAIL6STFAAHACENAAA
SCHEMBL27101416 0.91 PPARA (0.47) PPARAIL6STFAAHACENAAA
SCHEMBL14314072 0.87 PPARA (0.54) PPARAIL6STFAAHNAAAIDH1
SCHEMBL13316517 0.87 PPARA (0.54) PPARAIL6STFAAHNAAAIDH1
SCHEMBL13378242 0.86 IL6ST (0.49) PPARAIL6STFAAHNAAAIDH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0966429-B1 VALNOCTAMIDE STEREOISOMERS, A METHOD FOR THEIR SYNTHESIS AND SEPARATION AND USES THEREOF YISSUM RES DEV CO (IL) 2003-06-04 EP disclosed
US-6417399-B1 ETHYLATION OF ISOLEUCINE TO 3-METHYLVALERIC ACID; HALOACYLATION TO METHYL VALEROYL CHLORIDE; CARBOXYLATION TO VALNOCTIC ACID; AMIDATION TO VALNOCTAMIDE; ANTIEPILEPTIC AGENTS; PSYCHOLOGICAL DISORDERS YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM (IL) 2002-07-09 US disclosed