SCHEMBL7135463

SCHEMBL7135463

COc1ccc(C(C)(C(F)(F)F)C(F)(F)F)cc1CN[C@H]1CCCN(C(=O)OC(C)(C)C)[C@H]1c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 15/20 0.51
CYP2D6 P10635 4/20 0.51
CFTR P13569 4/20 0.45
KCNH2 Q12809 1/20 0.42
HTR1A P08908 1/20 0.42
HTR2A P28223 1/20 0.42
HTR2C P28335 1/20 0.42
HRH1 P35367 1/20 0.42
HTR2B P41595 1/20 0.42
SLC6A3 Q01959 1/20 0.42
TMEM97 Q5BJF2 1/20 0.42
SIGMAR1 Q99720 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8708427 1.00 TACR1 (0.51) TACR1CYP2D6CFTRKCNH2HTR1A
SCHEMBL7133654 0.94 TACR1 (0.60) TACR1CYP2D6CFTRKCNH2HTR1A
SCHEMBL7867202 0.94 TACR1 (0.60) TACR1CYP2D6CFTRKCNH2HTR1A
SCHEMBL7137909 0.94 TACR1 (0.51) TACR1CYP2D6CFTRKCNH2HTR1A
SCHEMBL7586407 0.90 TACR1 (0.48) TACR1CYP2D6CFTRKCNH2HTR1A
SCHEMBL7594455 0.89 TACR1 (0.50) TACR1CYP2D6CFTR
SCHEMBL7594451 0.89 TACR1 (0.50) TACR1CYP2D6CFTR
SCHEMBL7139592 0.89 TACR1 (0.47) TACR1CYP2D6CFTRKCNH2HTR1A
SCHEMBL7867174 0.89 TACR1 (0.47) TACR1CYP2D6CFTRKCNH2HTR1A
SCHEMBL7591379 0.89 TACR1 (0.49) TACR1CYP2D6CFTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6506775-B1 Treatment of a gastrointestinal disorder; a central nervous system (CNS) adverse conditions caused by Heliobacter pylori; or angiogenesis especially CNS disorders in a mammalian subject, especially humans. PFIZER INC 2003-01-14 US disclosed