SCHEMBL7148313

SCHEMBL7148313

CC(c1ncc(-n2ccnc2)c(-c2ccc(Cl)cc2Cl)n1)c1ccccc1N

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 1/20 0.46
GSK3A P49840 1/20 0.46
GSK3B P49841 1/20 0.46
IDO1 P14902 3/20 0.45
CNR1 P21554 1/20 0.40
CNR2 P34972 1/20 0.40
IDH1 O75874 2/20 0.36
CYP19A1 P11511 1/20 0.35
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
HSP90AB1 P08238 1/20 0.35
DPP4 P27487 1/20 0.34
BDKRB2 P30411 1/20 0.34
FBP1 P09467 1/20 0.34
ADRA2C P18825 1/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5089674 0.85 CDK1 (0.48) CDK1GSK3AGSK3BIDO1CNR1
SCHEMBL27253612 0.77 CDK1 (0.49) CDK1GSK3AGSK3BIDO1CNR1
SCHEMBL27538053 0.74 GSK3B (0.56) CDK1GSK3AGSK3BIDO1CNR1
SCHEMBL27559817 0.73 IDO1 (0.55) CDK1GSK3AGSK3BIDO1CNR1
SCHEMBL5089665 0.73 CDK1 (0.51) CDK1GSK3AGSK3BIDO1CNR1
SCHEMBL5089661 0.72 GSK3B (0.60) CDK1GSK3AGSK3BIDO1CNR1
SCHEMBL5099510 0.71 CNR1 (0.51) CDK1GSK3AGSK3BIDO1CNR1
SCHEMBL29367195 0.71 IDO1 (0.50) CDK1GSK3AGSK3BIDO1CNR1
SCHEMBL7148319 0.70 GSK3B (0.50) CDK1GSK3AGSK3BIDO1CNR1
SCHEMBL802729 0.67 CDK1 (0.47) CDK1GSK3AGSK3BIDO1CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1317433-A2 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 2003-06-11 EP disclosed
WO-2002020495-A2 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 2002-03-14 WO disclosed