SCHEMBL7149141

SCHEMBL7149141

COCN1c2cc(Cn3cnc(C=C(C)C(=O)O)c3)ccc2Sc2nccnc21

nearest known ligand 0.37

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 2/20 0.37
TBXAS1 P24557 3/20 0.35
ICAM1 P05362 4/20 0.35
CLK1 P49759 3/20 0.32
DYRK1A Q13627 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6745900 0.87 HDAC6 (0.37) HDAC6TBXAS1ICAM1CLK1DYRK1A
SCHEMBL6745906 0.87 HDAC6 (0.37) HDAC6TBXAS1ICAM1CLK1DYRK1A
SCHEMBL6750198 0.82 HDAC6 (0.36) HDAC6TBXAS1ICAM1CLK1DYRK1A
SCHEMBL6750191 0.82 HDAC6 (0.36) HDAC6TBXAS1ICAM1CLK1DYRK1A
SCHEMBL6750296 0.78 HDAC6 (0.42) HDAC6
SCHEMBL6745730 0.78 HDAC6 (0.43) HDAC6ICAM1
SCHEMBL6747454 0.77 HDAC6 (0.43) HDAC6ICAM1CLK1DYRK1A
SCHEMBL6747321 0.76 CYP11B1 (0.34) HDAC6
SCHEMBL6747445 0.76 HDAC6 (0.39) HDAC6ICAM1
SCHEMBL6749766 0.76 HDAC6 (0.40) HDAC6ICAM1CLK1DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6518423-B1 These compounds are useful as drugs efficacious in the prevention and treatment of these various inflammatory diseases and immunologic diseases, such as rheumatoid arthritis, atopic dermatitis, psoriasis, asthma, and EISAI CO., LTD. (JP) 2003-02-11 US disclosed