SCHEMBL7155282

SCHEMBL7155282

O=C1c2cccc(Sc3ccc(O)cc3)c2C(=O)c2c(Sc3ccc(O)cc3)cccc21

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.72
MAPK1 P28482 3/20 0.72
KDM4E B2RXH2 2/20 0.72
NSD2 O96028 1/20 0.72
P4HB P07237 4/20 0.50
ALDH1A1 P00352 3/20 0.48
MAOA P21397 2/20 0.48
TSHR P16473 2/20 0.48
TDP1 Q9NUW8 2/20 0.48
LMNA P02545 1/20 0.48
HPGD P15428 1/20 0.48
ALOX15 P16050 1/20 0.48
MAOB P27338 1/20 0.48
HTT P42858 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
HSD17B10 Q99714 1/20 0.48
NR1H2 P55055 1/20 0.43
DHFR P00374 1/20 0.40
BACE1 P56817 1/20 0.40
ELANE P08246 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6821902 0.95 MAPT (0.64) MAPTMAPK1KDM4ENSD2P4HB
SCHEMBL8441887 0.93 MAPT (0.68) MAPTMAPK1KDM4ENSD2P4HB
SCHEMBL8583274 0.89 MAPT (0.71) MAPTMAPK1KDM4ENSD2P4HB
SCHEMBL29365916 0.84 MAPT (1.00) MAPTMAPK1KDM4ENSD2ALDH1A1
SCHEMBL3459973 0.84 MAPT (1.00) MAPTMAPK1KDM4ENSD2ALDH1A1
SCHEMBL17284185 0.83 MAPK1 (0.72) MAPTMAPK1KDM4ENSD2ALDH1A1
SCHEMBL9581277 0.81 ADORA2A (0.51) MAPTMAPK1KDM4ENSD2P4HB
Anthraquinone SCHEMBL11411972 0.79 MAPT (0.89) MAPTMAPK1KDM4ENSD2ALDH1A1
SCHEMBL30475313 0.79 MAPT (0.89) MAPTMAPK1KDM4ENSD2ALDH1A1
SCHEMBL285567 0.79 MAPT (0.89) MAPTMAPK1KDM4ENSD2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3145997-B1 POLYMERIZABLE DICHROIC DYES ROLIC TECH AG (CH) 2023-07-12 EP disclosed
US-10385215-B2 Polymerizable dichroic dyes ROLIC AG (CH) 2019-08-20 US disclosed
US-20170058126-A1 POLYMERIZABLE DICHROIC DYES ROLIC AG (CH) 2017-03-02 US disclosed
US-20170058126-A1 POLYMERIZABLE DICHROIC DYES ROLIC AG (CH) 2017-03-02 US disclosed
WO-2015177062-A1 POLYMERIZABLE DICHROIC DYES ROLIC AG (CH) 2015-11-26 WO disclosed
EP-0797638-B1 ERASABLE INK COMPOSITION AND MARKING INSTRUMENT CONTAINING SAME BIC CORP (US) 2003-06-04 EP disclosed
US-5852072-A Erasable ink composition containing a waterborne polyurethane urea BIC CORPORATION (US) 1998-12-22 US disclosed
EP-0797638-A1 ERASABLE INK COMPOSITION AND MARKING INSTRUMENT CONTAINING SAME BIC CORPORATION (US) 1997-10-01 EP disclosed
WO-1996018697-A1 ERASABLE INK COMPOSITION AND MARKING INSTRUMENT CONTAINING SAME BIC CORPORATION (US) 1996-06-20 WO disclosed