SCHEMBL7156641

SCHEMBL7156641

C[C@H](NC(=O)C(O)c1cc(F)cc(F)c1)C(=O)NC1CN(c2ccccc2)c2ccccc2NC1C=O

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 13/20 0.47
PSEN2 P49810 13/20 0.47
APH1B Q8WW43 13/20 0.47
NCSTN Q92542 13/20 0.47
APH1A Q96BI3 13/20 0.47
PSENEN Q9NZ42 13/20 0.47
SPPL2A Q8TCT8 1/20 0.47
GSAP A4D1B5 1/20 0.32
GRM7 Q14831 1/20 0.31
MAPT P10636 1/20 0.31
EIF2S1 P05198 2/20 0.31
EIF2AK3 Q9NZJ5 2/20 0.31
MTNR1A P48039 1/20 0.30
MTNR1B P49286 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4986437 0.77 PSEN1 (0.61) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL4412059 0.69 PSEN1 (0.71) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL4419147 0.69 PSEN1 (0.80) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL21730143 0.67 PSEN1 (0.68) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL4841492 0.65 PSEN1 (0.53) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL4838006 0.65 PSEN1 (0.53) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL4842341 0.65 PSEN1 (0.53) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL4841306 0.65 PSEN1 (0.53) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL4844991 0.65 PSEN1 (0.47) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL4841555 0.65 PSEN1 (0.47) PSEN1PSEN2APH1BNCSTNAPH1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6544978-B2 Treating Alzheimer's disease both prophylactically and therapeutically ATHENA NEUROSCIENCES, INC. 2003-04-08 US disclosed