SCHEMBL7160352

SCHEMBL7160352

O=C1NCCn2c(-c3ccc(CN4CCc5ccccc5C4)cc3)nc3cccc1c32

nearest known ligand 0.66

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 20/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7162182 0.85 PARP1 (0.76) PARP1
SCHEMBL6198078 0.84 PARP1 (0.74) PARP1
SCHEMBL12750713 0.84 PARP1 (0.61) PARP1
SCHEMBL6202025 0.83 PARP1 (0.71) PARP1
SCHEMBL5076311 0.83 PARP1 (0.71) PARP1
SCHEMBL6200103 0.82 PARP1 (0.80) PARP1
SCHEMBL7160503 0.81 PARP1 (0.75) PARP1
SCHEMBL7156708 0.81 PARP1 (0.81) PARP1
SCHEMBL7161547 0.81 PARP1 (0.74) PARP1
SCHEMBL7161036 0.80 PARP1 (0.70) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6548494-B1 3,4-dihydro-2H-(1,4)diazepino(6,7,1-hi)indol-1-one or 1-thione derivatives where indole C3 could also be N; use treating cancers as well as stroke, head trauma, and neurodegenerative diseases AGOURON PHARMACEUTICALS, INC. 2003-04-15 US disclosed