SCHEMBL7166209

SCHEMBL7166209

O=C(Nc1nc2c(O)ccc(N3CCOCC3)c2s1)c1ccc(CCl)cc1.O=C(Nc1nc2c(OCc3ccccc3)ccc(N3CCOCC3)c2s1)c1ccc(CCl)cc1

nearest known ligand 0.46

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 17/20 0.46
ADORA1 P30542 13/20 0.46
ADORA2B P29275 3/20 0.45
WNT3A P56704 1/20 0.45
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
ADORA3 P0DMS8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3049798 0.96 ADORA2A (0.49) ADORA2AADORA1ADORA2BWNT3AMEN1
SCHEMBL3053434 0.89 LRRK2 (0.47) ADORA2AADORA1ADORA2BMEN1KMT2A
SCHEMBL3048781 0.85 ADORA2A (0.46) ADORA2AADORA1ADORA2BWNT3AMEN1
SCHEMBL3044761 0.84 ADORA2A (0.64) ADORA2AADORA1ADORA2BMEN1KMT2A
SCHEMBL7147830 0.83 ADORA2A (0.59) ADORA2AADORA1ADORA2BMEN1KMT2A
SCHEMBL3049478 0.82 LRRK2 (0.53) ADORA2AADORA1ADORA2BMEN1KMT2A
SCHEMBL3044476 0.82 ADORA2A (0.48) ADORA2AADORA1ADORA2BMEN1KMT2A
SCHEMBL3053641 0.79 ADORA2A (0.64) ADORA2AADORA1ADORA2BMEN1KMT2A
SCHEMBL3058336 0.78 ADORA2A (0.60) ADORA2AADORA1ADORA2BADORA3
SCHEMBL3047856 0.77 ADORA2A (0.69) ADORA2AADORA1ADORA2BMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1303272-A2 BENZOTHIAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2003-04-23 EP disclosed
WO-2001097786-A2 BENZOTHIAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2001-12-27 WO disclosed