SCHEMBL7167244

SCHEMBL7167244

CC1C(NC(=O)c2cnc(-c3cccc(F)c3F)s2)C2CCN1CC2

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 15/20 0.39
CHRNB2 P17787 9/20 0.39
CHRNA4 P43681 9/20 0.39
HTR3A P46098 2/20 0.38
USP30 Q70CQ3 1/20 0.37
MAPK11 Q15759 1/20 0.36
MAPK14 Q16539 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7120479 1.00 CHRNA7 (0.39) CHRNA7CHRNB2CHRNA4HTR3AUSP30
SCHEMBL7122228 0.93 CHRNA7 (0.41) CHRNA7CHRNB2CHRNA4HTR3AUSP30
SCHEMBL7116924 0.89 CHRNA7 (0.41) CHRNA7CHRNB2CHRNA4HTR3AUSP30
SCHEMBL7224711 0.86 CHRNA7 (0.42) CHRNA7CHRNB2CHRNA4USP30
SCHEMBL7114479 0.85 USP30 (0.41) CHRNA7CHRNB2CHRNA4HTR3AUSP30
SCHEMBL7112823 0.85 USP30 (0.41) CHRNA7CHRNB2CHRNA4HTR3AUSP30
SCHEMBL7130507 0.85 MAPK11 (0.45) CHRNA7CHRNB2CHRNA4HTR3AUSP30
SCHEMBL7129596 0.85 CHRNA7 (0.42) CHRNA7CHRNB2CHRNA4
SCHEMBL7114708 0.85 PIM1 (0.38) CHRNA7CHRNB2CHRNA4HTR3A
SCHEMBL7129282 0.85 HDAC3 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1311505-A2 QUINUCLIDINE-SUBSTITUTED HETEROARYL MOIETIES FOR TREATMENT OF DISEASE ( NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS ) PHARMACIA & UPJOHN COMPANY (US) 2003-05-21 EP claimed
WO-2002016355-A2 QUINUCLIDINE-SUBSTITUTED HETEROARYL MOIETIES FOR TREATMENT OF DISEASE (NICOTINIC) ACETYLCHOLINE RECEPTOR LIGANDS PHARMACIA & UPJOHN COMPANY (US) 2002-02-28 WO claimed