SCHEMBL7168231

SCHEMBL7168231

O=C(O)c1cc2c(OCc3ccccc3)cc(OCc3ccccc3)cc2[nH]1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 3/20 0.72
ALDH1A1 P00352 3/20 0.61
HPGD P15428 3/20 0.61
KDM4E B2RXH2 2/20 0.61
CYP1A2 P05177 2/20 0.61
HSD17B10 Q99714 2/20 0.61
CYP2C9 P11712 1/20 0.61
SRD5A1 P18405 1/20 0.56
MEN1 O00255 2/20 0.55
KMT2A Q03164 2/20 0.55
IDO1 P14902 1/20 0.49
TDO2 P48775 1/20 0.49
RHEB Q15382 2/20 0.49
CTSV O60911 1/20 0.49
CTSL P07711 1/20 0.49
PDGFRB P09619 1/20 0.48
PDGFRA P16234 1/20 0.48
MDH2 P40926 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
NR4A2 P43354 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30169467 1.00 SRD5A2 (0.72) SRD5A2ALDH1A1HPGDKDM4ECYP1A2
SCHEMBL30396449 0.91 SRD5A2 (0.64) SRD5A2ALDH1A1HPGDKDM4ECYP1A2
SCHEMBL7197823 0.91 SRD5A2 (0.67) SRD5A2ALDH1A1HPGDKDM4ECYP1A2
SCHEMBL28594443 0.89 SRD5A2 (0.61) SRD5A2ALDH1A1HPGDKDM4ECYP1A2
SCHEMBL28581075 0.89 SRD5A2 (0.65) SRD5A2ALDH1A1HPGDKDM4ECYP1A2
SCHEMBL28917192 0.88 SRD5A2 (0.63) SRD5A2ALDH1A1HPGDKDM4ECYP1A2
SCHEMBL28586036 0.88 SRD5A2 (0.60) SRD5A2ALDH1A1HPGDKDM4ECYP1A2
SCHEMBL7168633 0.88 SRD5A2 (0.56) SRD5A2ALDH1A1HPGDKDM4ECYP1A2
Dimethylamine SCHEMBL28585893 0.86 SRD5A2 (0.61) SRD5A2ALDH1A1HPGDKDM4ECYP1A2
Dimethylamine SCHEMBL28585501 0.86 SRD5A2 (0.58) SRD5A2ALDH1A1HPGDKDM4ECYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112358435-B Substituted aromatic heterocyclic compound, preparation method, ULK1 inhibition and antitumor application 中国医学科学院医药生物技术研究所 2023-01-10 CN disclosed
CN-112358435-A Substituted aromatic heterocyclic compound, preparation method, ULK1 inhibition and antitumor application 中国医学科学院医药生物技术研究所 2021-02-12 CN disclosed
EP-1328514-A1 AMIDE DERIVATIVES AS NMDA RECEPTOR ANTAGONISTS RICHTER GEDEON VEGYESZETI GYAR R.T. (HU) 2003-07-23 EP disclosed
WO-2002034718-A1 AMIDE DERIVATIVES AS NMDA RECEPTOR ANTAGONISTS RICHTER GEDEON VEGYESZETI GYAR RT. (HU) 2002-05-02 WO disclosed