SCHEMBL7173306

SCHEMBL7173306

COc1ccc(CNc2nc(Cl)nc3sc(C)c(C)c23)cc1OC.Cc1sc2nc(Cl)nc(Cl)c2c1C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.44
GAA P10253 2/20 0.44
CHRM4 P08173 1/20 0.44
RXFP1 Q9HBX9 1/20 0.44
TSHR P16473 1/20 0.43
TNF P01375 1/20 0.43
NOD1 Q9Y239 1/20 0.43
BCHE P06276 2/20 0.42
ACHE P22303 2/20 0.42
STAT1 P42224 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
APP P05067 3/20 0.41
POLB P06746 1/20 0.41
PDE5A O76074 1/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5129494 0.96 ESR1 (0.47) ESR1GAACHRM4RXFP1TSHR
SCHEMBL7171683 0.93 PDE5A (0.46) ESR1GAACHRM4RXFP1PDE5A
SCHEMBL7176322 0.90 TSHR (0.45) ESR1GAACHRM4TSHRTNF
SCHEMBL5130592 0.89 BCDIN3D (0.48) ESR1GAACHRM4RXFP1PDE5A
SCHEMBL5131031 0.87 TSHR (0.48) ESR1GAACHRM4TSHRTNF
SCHEMBL7175621 0.85 GAA (0.47) ESR1GAARXFP1LMNASMN1; SMN2
SCHEMBL7176456 0.83 PDE5A (0.46) ESR1CHRM4PDE5A
SCHEMBL7167188 0.82 GAA (0.50) ESR1GAACHRM4RXFP1LMNA
SCHEMBL7513169 0.82 CHRM4 (0.40) GAACHRM4RXFP1TSHRTNF
SCHEMBL5808228 0.82 POLB (0.44) CHRM4TNFNOD1BCHEACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0920431-B1 THIENOPYRIMIDINES MERCK PATENT GMBH (DE) 2003-02-26 EP disclosed