SCHEMBL7174648

SCHEMBL7174648

CCCCN(C(=O)c1cc(C)cc(C(N)=O)c1)[C@@H](Cc1cc(F)cc(F)c1)[C@H](O)CNCc1cccc(CC)c1

nearest known ligand 0.65

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.65
CTSD P07339 3/20 0.65
BACE2 Q9Y5Z0 3/20 0.53
CTSB P07858 6/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7608357 0.92 BACE1 (0.66) BACE1CTSDBACE2CTSB
SCHEMBL5343242 0.91 BACE1 (0.65) BACE1CTSDBACE2CTSB
SCHEMBL7672775 0.90 BACE1 (0.61) BACE1CTSDBACE2CTSB
SCHEMBL5436485 0.86 BACE1 (0.63) BACE1CTSDBACE2CTSB
SCHEMBL5378221 0.86 BACE1 (0.62) BACE1CTSDBACE2CTSB
SCHEMBL5369408 0.82 BACE1 (0.77) BACE1CTSDBACE2
SCHEMBL7608365 0.81 BACE1 (0.64) BACE1CTSDBACE2CTSB
SCHEMBL5388283 0.80 BACE1 (0.91) BACE1CTSDBACE2
SCHEMBL5351506 0.80 BACE1 (0.81) BACE1CTSDBACE2CTSB
SCHEMBL7613103 0.80 BACE1 (0.60) BACE1CTSDBACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2004502669-A 2004-01-29 JP claimed
EP-1353898-A2 COMPOUNDS TO TREAT ALZHEIMER'S DISEASE Elan Pharmaceuticals, Inc. (US) 2003-10-22 EP claimed
WO-2002002512-A2 COMPOUNDS TO TREAT ALZHEIMER'S DISEASE ELAN PHARMACEUTICALS, INC. (US) 2002-01-10 WO claimed