SCHEMBL717772

SCHEMBL717772

Cn1nccc1C1CCCN1C(=O)c1cccc(C(=O)N[C@@H](Cc2ccccc2)[C@H](O)CNCc2cccc(C(F)(F)F)c2)c1

nearest known ligand 0.55

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.55
CTSD P07339 19/20 0.55
BACE2 Q9Y5Z0 19/20 0.55
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL166486 1.00 BACE1 (0.55) BACE1CTSDBACE2CYP3A4CYP2D6
SCHEMBL164455 0.88 BACE1 (0.58) BACE1CTSDBACE2CYP3A4CYP2D6
SCHEMBL718496 0.88 BACE1 (0.58) BACE1CTSDBACE2CYP3A4CYP2D6
SCHEMBL719138 0.88 BACE1 (0.58) BACE1CTSDBACE2CYP3A4CYP2D6
SCHEMBL717347 0.88 BACE1 (0.58) BACE1CTSDBACE2CYP3A4CYP2D6
SCHEMBL166622 0.88 BACE1 (0.58) BACE1CTSDBACE2CYP3A4CYP2D6
SCHEMBL717348 0.88 BACE1 (0.58) BACE1CTSDBACE2CYP3A4CYP2D6
SCHEMBL166324 0.88 BACE1 (0.60) BACE1CTSDBACE2CYP3A4CYP2D6
SCHEMBL717774 0.88 BACE1 (0.60) BACE1CTSDBACE2CYP3A4CYP2D6
SCHEMBL175112 0.87 BACE1 (0.54) BACE1CTSDBACE2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120053200-A1 BACE 2 INHIBITORS HOFFMANN-LA ROCHE INC. 2012-03-01 US claimed
US-20120053200-A1 BACE 2 INHIBITORS HOFFMANN-LA ROCHE INC. 2012-03-01 US disclosed
US-20120053200-A1 BACE 2 INHIBITORS HOFFMANN-LA ROCHE INC. 2012-03-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120053200-A1 BACE 2 INHIBITORS BACE2, BACE1, PSEN2 BACE1 2/4885CTSD 138/4885BACE2 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.