SCHEMBL7181698

SCHEMBL7181698

COc1ccc(N2CCOCC2)c2sc(NC(=O)c3ccc(C(C)N)cc3)nc12

nearest known ligand 0.66

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 18/20 0.66
ADORA1 P30542 12/20 0.66
MEN1 O00255 1/20 0.60
KMT2A Q03164 1/20 0.60
ADORA2B P29275 4/20 0.59
ADORA3 P0DMS8 2/20 0.59
MAPT P10636 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3047230 0.91 ADORA2A (0.63) ADORA2AADORA1MEN1KMT2AADORA2B
SCHEMBL7185374 0.90 ADORA2A (0.62) ADORA2AADORA1ADORA2BADORA3
SCHEMBL5713454 0.89 ADORA2A (0.59) ADORA2AADORA1MEN1KMT2AADORA2B
SCHEMBL3052290 0.89 ADORA2A (0.65) ADORA2AADORA1MEN1KMT2AADORA2B
SCHEMBL28412423 0.88 ADORA2A (0.68) ADORA2AADORA1MEN1KMT2AADORA2B
SCHEMBL28416866 0.88 ADORA2A (0.68) ADORA2AADORA1MEN1KMT2AADORA2B
SCHEMBL3054173 0.87 ADORA2A (0.74) ADORA2AADORA1MEN1KMT2AADORA2B
SCHEMBL3047856 0.87 ADORA2A (0.69) ADORA2AADORA1MEN1KMT2AADORA2B
SCHEMBL3047910 0.87 ADORA2A (0.58) ADORA2AADORA1MEN1KMT2AADORA2B
SCHEMBL5713516 0.86 ADORA2A (0.64) ADORA2AADORA1MEN1KMT2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6521754-B2 Such as N-4-methoxy-7-morpholin-4-yl-benzothiazol-2-yl)-2-methyl-isoni cotinamide HOFFMAN-LA ROCHE INC. 2003-02-18 US disclosed