SCHEMBL7183653

SCHEMBL7183653

COc1cccc(-c2ccc3cc(OC)ccc3c2Oc2ccc(CCC(=O)O)cc2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 13/20 0.51
VDR P11473 1/20 0.50
PPARD Q03181 1/20 0.50
FFAR4 Q5NUL3 5/20 0.47
THRA P10827 1/20 0.46
THRB P10828 1/20 0.46
DGAT2 Q96PD7 1/20 0.45
KDM4E B2RXH2 1/20 0.44
NPC1 O15118 1/20 0.44
LMNA P02545 1/20 0.44
TP53 P04637 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
MAPT P10636 1/20 0.44
MAOA P21397 1/20 0.44
SLC6A2 P23975 1/20 0.44
RAB9A P51151 1/20 0.44
SLC6A3 Q01959 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
RXRA P19793 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7185982 0.94 FFAR1 (0.50) FFAR1VDRPPARDFFAR4THRA
SCHEMBL7181091 0.93 ESR1 (0.48) FFAR1VDRPPARDFFAR4
SCHEMBL7183920 0.93 FFAR1 (0.50) FFAR1VDRPPARDFFAR4THRA
SCHEMBL7187977 0.92 ESR1 (0.47) FFAR1VDRPPARDFFAR4LMNA
SCHEMBL7183632 0.90 FFAR1 (0.52) FFAR1FFAR4KDM4ENPC1LMNA
SCHEMBL7194279 0.88 CYP1A2 (0.47) FFAR1VDRPPARDTHRATHRB
SCHEMBL7187874 0.88 ESR1 (0.55) FFAR1FFAR4KDM4ENPC1LMNA
SCHEMBL7194015 0.87 FFAR1 (0.53) FFAR1FFAR4KDM4ENPC1LMNA
SCHEMBL7183696 0.87 FFAR1 (0.51) FFAR1FFAR4KDM4ENPC1LMNA
SCHEMBL7193901 0.86 MAPT (0.45) FFAR1VDRPPARDFFAR4THRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0835867-B1 1-Aryloxy-2-arylnaphthyl compounds, intermediates, compositions, and methods LILLY CO ELI (US) 2003-12-03 EP claimed
US-5916916-A USEFUL AS SELECTIVE ESTROGEN RECEPTOR MODULATORS. ELI LILLY AND COMPANY (US) 1999-06-29 US claimed
EP-0835867-A1 1-Aryloxy-2-arylnaphthyl compounds, intermediates, compositions, and methods ELI LILLY AND COMPANY (US) 1998-04-15 EP claimed
EP-0835867-B1 1-Aryloxy-2-arylnaphthyl compounds, intermediates, compositions, and methods LILLY CO ELI (US) 2003-12-03 EP disclosed
US-5916916-A USEFUL AS SELECTIVE ESTROGEN RECEPTOR MODULATORS. ELI LILLY AND COMPANY (US) 1999-06-29 US disclosed
EP-0835867-A1 1-Aryloxy-2-arylnaphthyl compounds, intermediates, compositions, and methods ELI LILLY AND COMPANY (US) 1998-04-15 EP disclosed