SCHEMBL7184366

SCHEMBL7184366

CC=CCc1cc(CC=CC)c(OCCC)c(C=CC(=O)c2ccc(NC)cc2)c1O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 2/20 0.40
DPP4 P27487 3/20 0.37
IDO1 P14902 1/20 0.36
CYP1A1 P04798 2/20 0.36
CYP1B1 Q16678 2/20 0.36
CYP3A4 P08684 2/20 0.35
TUBB4A P04350 2/20 0.33
TUBB P07437 2/20 0.33
TUBA3C P0DPH7 2/20 0.33
TUBA1B P68363 2/20 0.33
TUBA4A P68366 2/20 0.33
TUBB4B P68371 2/20 0.33
TUBB3 Q13509 2/20 0.33
TUBB2A Q13885 2/20 0.33
TUBB8 Q3ZCM7 2/20 0.33
TUBA3E Q6PEY2 2/20 0.33
TUBA1A Q71U36 2/20 0.33
TUBA1C Q9BQE3 2/20 0.33
TUBB6 Q9BUF5 2/20 0.33
TUBB2B Q9BVA1 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7184362 1.00 ABCG2 (0.40) ABCG2DPP4IDO1CYP1A1CYP1B1
SCHEMBL7184657 0.92 MAOB (0.38) ABCG2CYP1A1CYP1B1CYP3A4LMNA
SCHEMBL7184653 0.92 MAOB (0.38) ABCG2CYP1A1CYP1B1CYP3A4LMNA
SCHEMBL7183521 0.90 ABCG2 (0.51) ABCG2DPP4CYP1A1CYP1B1LMNA
SCHEMBL7183518 0.90 ABCG2 (0.51) ABCG2DPP4CYP1A1CYP1B1LMNA
SCHEMBL7189364 0.89 PTPN1 (0.42) ABCG2DPP4
SCHEMBL7189361 0.89 PTPN1 (0.42) ABCG2DPP4
SCHEMBL7186612 0.89 ABCG2 (0.42) ABCG2DPP4CYP1A1CYP1B1CYP3A4
SCHEMBL7186614 0.89 ABCG2 (0.42) ABCG2DPP4CYP1A1CYP1B1CYP3A4
SCHEMBL7190226 0.89 ABCG2 (0.42) ABCG2DPP4CYP1A1CYP1B1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6603046-B1 The invention is drawn to novel bis-aromatic a, beta -unsaturated ketones. The compounds are useful in the treatment and prophylaxis of diseases caused by parasites or bacteria. LICA PHARMACEUTICALS A/S (DK) 2003-08-05 US disclosed
EP-0634927-B1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES, OR BACTERIA LICA PHARMACEUTICALS AS (DK) 2001-07-04 EP disclosed
US-5985935-A PARASITICIDES OR BACTERICIDES STATENS SERUMINSTITUT (DK) 1999-11-16 US disclosed