SCHEMBL7186566

SCHEMBL7186566

CCOc1c(C)cc(C)c(O)c1/C=C/C(=O)c1ccc(O)cc1

nearest known ligand 0.55

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 4/20 0.55
MAOB P27338 3/20 0.55
POLB P06746 2/20 0.47
LMNA P02545 1/20 0.47
MAPT P10636 1/20 0.46
MAOA P21397 1/20 0.46
RAB9A P51151 1/20 0.46
CYP1A1 P04798 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP1B1 Q16678 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7186568 1.00 ABCG2 (0.55) ABCG2MAOBPOLBLMNAMAPT
SCHEMBL7179998 0.90 ABCG2 (0.57) ABCG2MAOBPOLBMAPTMAOA
SCHEMBL7179996 0.90 ABCG2 (0.57) ABCG2MAOBPOLBMAPTMAOA
SCHEMBL7185365 0.90 CA1 (0.46) ABCG2MAOBCYP1A1CYP1A2CYP2D6
SCHEMBL7185369 0.90 CA1 (0.46) ABCG2MAOBCYP1A1CYP1A2CYP2D6
SCHEMBL7180061 0.89 MAOB (0.43) ABCG2MAOBMAPTRAB9ACYP1A1
SCHEMBL7180055 0.89 MAOB (0.43) ABCG2MAOBMAPTRAB9ACYP1A1
SCHEMBL9203705 0.85 MAOB (0.42) ABCG2MAOBPOLBLMNAMAPT
SCHEMBL9203700 0.85 MAOB (0.42) ABCG2MAOBPOLBLMNAMAPT
SCHEMBL7192207 0.85 MAPT (0.46) ABCG2MAOBPOLBMAPTMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6603046-B1 The invention is drawn to novel bis-aromatic a, beta -unsaturated ketones. The compounds are useful in the treatment and prophylaxis of diseases caused by parasites or bacteria. LICA PHARMACEUTICALS A/S (DK) 2003-08-05 US disclosed
EP-0634927-B1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES, OR BACTERIA LICA PHARMACEUTICALS AS (DK) 2001-07-04 EP disclosed
US-5985935-A PARASITICIDES OR BACTERICIDES STATENS SERUMINSTITUT (DK) 1999-11-16 US disclosed