SCHEMBL7187702

SCHEMBL7187702

CCCc1ccc(OCC)c(/C=C/C(=O)c2ccc(O)cc2)c1OCC

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 4/20 0.51
MAOB P27338 2/20 0.51
LMNA P02545 4/20 0.49
POLB P06746 1/20 0.49
CYP1A1 P04798 2/20 0.45
CYP1A2 P05177 2/20 0.45
CYP2D6 P10635 2/20 0.45
CYP1B1 Q16678 2/20 0.45
CAPN1 P07384 1/20 0.43
MAPT P10636 4/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
ATM Q13315 1/20 0.43
PDE4A P27815 1/20 0.42
PDE4B Q07343 1/20 0.42
PDE4C Q08493 1/20 0.42
PDE4D Q08499 1/20 0.42
KDM4E B2RXH2 2/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
ALDH1A1 P00352 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7187705 1.00 ABCG2 (0.51) ABCG2MAOBLMNAPOLBCYP1A1
SCHEMBL7183455 0.90 CYP1B1 (0.44) ABCG2MAOBLMNAPOLBCYP1A1
SCHEMBL7183451 0.90 CYP1B1 (0.44) ABCG2MAOBLMNAPOLBCYP1A1
SCHEMBL7179925 0.90 ABCG2 (0.54) ABCG2MAOBLMNAPOLBCYP1A1
SCHEMBL7187779 0.89 ABCG2 (0.56) ABCG2MAOBLMNAPOLBCYP1A2
SCHEMBL8469442 0.89 ABCG2 (0.56) ABCG2MAOBLMNAPOLBCYP1A2
SCHEMBL7184677 0.88 MAPT (0.44) ABCG2MAOBLMNAPOLBCYP1A1
SCHEMBL7177798 0.88 CYP1A1 (0.42) ABCG2MAOBLMNAPOLBCYP1A1
SCHEMBL7177791 0.88 CYP1A1 (0.42) ABCG2MAOBLMNAPOLBCYP1A1
SCHEMBL7184673 0.88 MAPT (0.44) ABCG2MAOBLMNAPOLBCYP1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6603046-B1 The invention is drawn to novel bis-aromatic a, beta -unsaturated ketones. The compounds are useful in the treatment and prophylaxis of diseases caused by parasites or bacteria. LICA PHARMACEUTICALS A/S (DK) 2003-08-05 US disclosed
EP-0634927-B1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES, OR BACTERIA LICA PHARMACEUTICALS AS (DK) 2001-07-04 EP disclosed
US-5985935-A PARASITICIDES OR BACTERICIDES STATENS SERUMINSTITUT (DK) 1999-11-16 US disclosed
EP-0634927-A1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES, OR BACTERIA STATENS SERUMINSTITUT (DK) 1995-01-25 EP disclosed
WO-1993017671-A1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES, OR BACTERIA STATENS SERUMINSTITUT (DK) 1993-09-16 WO disclosed