SCHEMBL7187829

SCHEMBL7187829

CCC(C)(C)c1cc(C(C)(C)CC)c(OC(=O)C(C)(C)C)c(/C=C/C(=O)c2ccc(OC(=O)C(C)(C)C)cc2)c1OC

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 6/20 0.43
MAPT P10636 4/20 0.43
LMNA P02545 2/20 0.43
ALDH1A1 P00352 2/20 0.43
KDM4E B2RXH2 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
ABCG2 Q9UNQ0 2/20 0.43
TNFRSF1A P19438 1/20 0.42
KRAS P01116 1/20 0.42
ELANE P08246 2/20 0.42
MAPK1 P28482 1/20 0.42
BCHE P06276 1/20 0.40
IDH1 O75874 1/20 0.40
ABCB1 P08183 1/20 0.40
UGT1A1 P22309 1/20 0.40
DPP4 P27487 1/20 0.40
ABCC1 P33527 1/20 0.40
PRMT6 Q96LA8 1/20 0.40
MAOB P27338 1/20 0.40
F3 P13726 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7187830 1.00 PTPN1 (0.43) PTPN1MAPTLMNAALDH1A1KDM4E
SCHEMBL7184517 0.91 MAOB (0.44) MAPTLMNAALDH1A1KDM4ESMN1; SMN2
SCHEMBL7184524 0.91 MAOB (0.44) MAPTLMNAALDH1A1KDM4ESMN1; SMN2
SCHEMBL7186734 0.89 TNFRSF1A (0.54) PTPN1MAPTLMNAALDH1A1ABCG2
SCHEMBL7186739 0.89 TNFRSF1A (0.54) PTPN1MAPTLMNAALDH1A1ABCG2
SCHEMBL7192597 0.89 ABCG2 (0.46) PTPN1MAPTLMNAALDH1A1KDM4E
SCHEMBL7185965 0.89 ELANE (0.40) PTPN1ABCG2ELANEBCHEMAOB
SCHEMBL7192600 0.89 ABCG2 (0.46) PTPN1MAPTLMNAALDH1A1KDM4E
SCHEMBL7185970 0.89 ELANE (0.40) PTPN1ABCG2ELANEBCHEMAOB
SCHEMBL7190988 0.88 PTPN1 (0.47) PTPN1MAPTLMNAALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6603046-B1 The invention is drawn to novel bis-aromatic a, beta -unsaturated ketones. The compounds are useful in the treatment and prophylaxis of diseases caused by parasites or bacteria. LICA PHARMACEUTICALS A/S (DK) 2003-08-05 US disclosed
EP-0634927-B1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES, OR BACTERIA LICA PHARMACEUTICALS AS (DK) 2001-07-04 EP disclosed
US-5985935-A PARASITICIDES OR BACTERICIDES STATENS SERUMINSTITUT (DK) 1999-11-16 US disclosed