SCHEMBL7187979

SCHEMBL7187979

CCCOc1ccc(C)c(OCCC)c1C=CC(=O)c1ccc(N)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.45
CA2 P00918 2/20 0.45
KRAS P01116 1/20 0.45
ABCG2 Q9UNQ0 3/20 0.44
GAA P10253 2/20 0.44
CYP1B1 Q16678 3/20 0.41
CYP1A1 P04798 2/20 0.41
CTSL P07711 1/20 0.41
CTSB P07858 1/20 0.41
DPP4 P27487 2/20 0.40
MEN1 O00255 2/20 0.40
ALDH1A1 P00352 2/20 0.40
MAPT P10636 2/20 0.40
HTT P42858 2/20 0.40
KMT2A Q03164 2/20 0.40
NPC1 O15118 1/20 0.40
LMNA P02545 1/20 0.40
NFKB1 P19838 1/20 0.40
RAB9A P51151 1/20 0.40
NFKB2 Q00653 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7180664 0.94 ABCG2 (0.46) CA1CA2KRASABCG2CYP1B1
SCHEMBL7184600 0.89 ABCG2 (0.57) ABCG2CYP1B1CYP1A1CTSLCTSB
SCHEMBL7177660 0.88 CYP1B1 (0.47) CA1CA2KRASABCG2CYP1B1
SCHEMBL7177657 0.88 CYP1B1 (0.47) CA1CA2KRASABCG2CYP1B1
SCHEMBL7181412 0.87 CA1 (0.43) CA1CA2KRASABCG2GAA
SCHEMBL7189584 0.86 CA1 (0.42) CA1CA2KRASABCG2GAA
SCHEMBL7184172 0.86 ABCG2 (0.43) ABCG2CYP1B1CYP1A1DPP4ALDH1A1
SCHEMBL7184017 0.86 ABCG2 (0.43) ABCG2CYP1B1CYP1A1DPP4MAPT
SCHEMBL7184853 0.85 ABCG2 (0.57) CA1CA2KRASABCG2GAA
SCHEMBL7190653 0.85 PTPN1 (0.41) CA1CA2KRASABCG2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6603046-B1 The invention is drawn to novel bis-aromatic a, beta -unsaturated ketones. The compounds are useful in the treatment and prophylaxis of diseases caused by parasites or bacteria. LICA PHARMACEUTICALS A/S (DK) 2003-08-05 US disclosed
EP-0634927-B1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES, OR BACTERIA LICA PHARMACEUTICALS AS (DK) 2001-07-04 EP disclosed
US-5985935-A PARASITICIDES OR BACTERICIDES STATENS SERUMINSTITUT (DK) 1999-11-16 US disclosed
EP-0634927-A1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES, OR BACTERIA STATENS SERUMINSTITUT (DK) 1995-01-25 EP disclosed
WO-1993017671-A1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES, OR BACTERIA STATENS SERUMINSTITUT (DK) 1993-09-16 WO disclosed