SCHEMBL7189059

SCHEMBL7189059

COc1cc(OC)c(C=CC(=O)c2ccc(N)cc2)cc1C

nearest known ligand 0.69

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 2/20 0.69
CTSL P07711 2/20 0.68
CTSB P07858 2/20 0.68
PTPN1 P18031 2/20 0.67
CA1 P00915 2/20 0.60
CA2 P00918 2/20 0.60
KRAS P01116 1/20 0.60
DPP4 P27487 4/20 0.57
SNCA P37840 2/20 0.56
CAPN1 P07384 1/20 0.56
TNFRSF1A P19438 1/20 0.56
TDP1 Q9NUW8 1/20 0.56
CYP1A1 P04798 2/20 0.53
CYP1B1 Q16678 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7189052 1.00 ABCG2 (0.69) ABCG2CTSLCTSBPTPN1CA1
SCHEMBL7101429 0.90 ABCG2 (0.85) ABCG2CTSLCTSBPTPN1CA1
SCHEMBL7184183 0.90 PTPN1 (0.76) ABCG2CTSLCTSBPTPN1CA1
SCHEMBL7184180 0.90 PTPN1 (0.76) ABCG2CTSLCTSBPTPN1CA1
SCHEMBL9111986 0.88 TNFRSF1A (0.72) ABCG2PTPN1KRASDPP4TNFRSF1A
SCHEMBL7184370 0.88 DPP4 (0.74) ABCG2CTSLCTSBPTPN1DPP4
SCHEMBL9111983 0.88 TNFRSF1A (0.72) ABCG2PTPN1KRASDPP4TNFRSF1A
SCHEMBL7184368 0.88 DPP4 (0.74) ABCG2CTSLCTSBPTPN1DPP4
SCHEMBL7178662 0.84 ABCG2 (0.66) ABCG2CTSLCTSBPTPN1DPP4
SCHEMBL7192010 0.84 ABCG2 (0.66) ABCG2CTSLCTSBPTPN1DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6603046-B1 The invention is drawn to novel bis-aromatic a, beta -unsaturated ketones. The compounds are useful in the treatment and prophylaxis of diseases caused by parasites or bacteria. LICA PHARMACEUTICALS A/S (DK) 2003-08-05 US disclosed
EP-0634927-B1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES, OR BACTERIA LICA PHARMACEUTICALS AS (DK) 2001-07-04 EP disclosed
US-5985935-A PARASITICIDES OR BACTERICIDES STATENS SERUMINSTITUT (DK) 1999-11-16 US disclosed
EP-0634927-A1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES, OR BACTERIA STATENS SERUMINSTITUT (DK) 1995-01-25 EP disclosed
WO-1993017671-A1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES, OR BACTERIA STATENS SERUMINSTITUT (DK) 1993-09-16 WO disclosed