SCHEMBL7190078

SCHEMBL7190078

COc1c(OC(C)C)c(C=CC(=O)c2ccc(OC(=O)C(C)(C)C)cc2)cc(C(C)C)c1OC(=O)C(C)(C)C

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 9/20 0.43
ABCG2 Q9UNQ0 3/20 0.41
GABRA3 P34903 1/20 0.40
GABRA2 P47869 1/20 0.40
GABRB2 P47870 1/20 0.40
TNFRSF1A P19438 1/20 0.40
CYP1A1 P04798 1/20 0.40
CYP1B1 Q16678 1/20 0.40
IDH1 O75874 1/20 0.40
ABCB1 P08183 1/20 0.40
UGT1A1 P22309 1/20 0.40
DPP4 P27487 1/20 0.40
ABCC1 P33527 1/20 0.40
PRMT6 Q96LA8 1/20 0.40
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
MAPK1 P28482 1/20 0.39
KRAS P01116 1/20 0.39
ELANE P08246 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7186746 0.94 PTPN1 (0.46) PTPN1ABCG2GABRA3GABRA2GABRB2
SCHEMBL9275539 0.90 TNFRSF1A (0.39) PTPN1ABCG2TNFRSF1ACYP1A1CYP1B1
SCHEMBL7191627 0.89 CYP1A1 (0.47) PTPN1ABCG2CYP1A1CYP1B1DPP4
SCHEMBL7189148 0.89 TNFRSF1A (0.47) PTPN1ABCG2GABRA3GABRA2GABRB2
SCHEMBL7188849 0.89 ELANE (0.40) PTPN1ABCG2CYP1A1CYP1B1IDH1
SCHEMBL7188844 0.89 ELANE (0.40) PTPN1ABCG2CYP1A1CYP1B1IDH1
SCHEMBL7187085 0.89 PTPN1 (0.43) PTPN1ABCG2GABRA3GABRA2GABRB2
SCHEMBL7191566 0.88 PTPN1 (0.44) PTPN1ABCG2GABRA3GABRA2GABRB2
SCHEMBL7191564 0.88 PTPN1 (0.44) PTPN1ABCG2GABRA3GABRA2GABRB2
SCHEMBL7190809 0.87 PTPN1 (0.44) PTPN1ABCG2GABRA3GABRA2GABRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6603046-B1 The invention is drawn to novel bis-aromatic a, beta -unsaturated ketones. The compounds are useful in the treatment and prophylaxis of diseases caused by parasites or bacteria. LICA PHARMACEUTICALS A/S (DK) 2003-08-05 US disclosed
EP-0634927-B1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES, OR BACTERIA LICA PHARMACEUTICALS AS (DK) 2001-07-04 EP disclosed