SCHEMBL7196006

SCHEMBL7196006

Cc1ccccc1C(=O)c1ccc(Nc2ccc(Br)cc2[N+](=O)[O-])cc1F

nearest known ligand 0.60

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPK13 O15264 10/20 0.60
MAPK12 P53778 10/20 0.60
MAPK11 Q15759 10/20 0.60
MAPK14 Q16539 10/20 0.60
ALDH3A1 P30838 1/20 0.48
LMNA P02545 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
ALDH1A1 P00352 1/20 0.44
ATM Q13315 1/20 0.44
MEN1 O00255 4/20 0.42
KMT2A Q03164 4/20 0.42
RAB9A P51151 1/20 0.42
GFER P55789 1/20 0.41
HCAR3 P49019 1/20 0.41
MAPT P10636 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7192088 0.88 MAPK13 (0.76) MAPK13MAPK12MAPK11MAPK14ALDH3A1
SCHEMBL7198829 0.88 MAPK14 (0.79) MAPK13MAPK12MAPK11MAPK14LMNA
SCHEMBL7198684 0.86 AKR1C3 (0.53) MAPK13MAPK12MAPK11MAPK14ALDH3A1
SCHEMBL5173305 0.86 MAPK13 (0.61) MAPK13MAPK12MAPK11MAPK14LMNA
SCHEMBL7195744 0.84 MAPK13 (0.56) MAPK13MAPK12MAPK11MAPK14LMNA
SCHEMBL6396818 0.83 MAPK14 (0.77) MAPK13MAPK12MAPK11MAPK14MEN1
SCHEMBL6907054 0.82 MAPK13 (0.57) MAPK13MAPK12MAPK11MAPK14LMNA
SCHEMBL7198676 0.80 MAPK13 (0.61) MAPK13MAPK12MAPK11MAPK14ALDH3A1
SCHEMBL7196494 0.80 MAPK14 (0.67) MAPK13MAPK12MAPK11MAPK14LMNA
SCHEMBL7196766 0.80 MAPK14 (0.79) MAPK13MAPK12MAPK11MAPK14ALDH3A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1202954-B1 NOVEL AMINOBENZOPHENONES LEO PHARMA AS (DK) 2003-10-01 EP disclosed
US-6624199-B1 Prophylaxis and treatment of acne and acne related skin diseases with aminobenzophenones, and novel compounds effective in the treatment, as well as pharmaceutical preparations containing these compounds and dosage units LEO PHARMACEUTICALS PRODUCTS LTD. A/S (DK) 2003-09-23 US disclosed
EP-1202954-A1 NOVEL AMINOBENZOPHENONES LEO PHARMACEUTICAL PRODUCTS LTD. A/S (LOVENS KEMISKE FABRIK PRODUKTIONSAKTIESELSKAB) (DK) 2002-05-08 EP disclosed
WO-2001005744-A1 NOVEL AMINOBENZOPHENONES Leo Pharmaceutical Products Ltd. A/S (Løvens Kemiske Fabrik Produktionsaktieselskab) (DK) 2001-01-25 WO disclosed