SCHEMBL7204709

SCHEMBL7204709

Nc1nc(N)c2nc(O)n(Cc3ccccc3)c2n1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.47
ADORA1 P30542 1/20 0.47
PTPRF P10586 1/20 0.46
PTPN1 P18031 1/20 0.46
PTPRA P18433 1/20 0.46
PTPN11 Q06124 1/20 0.46
TLR7 Q9NYK1 11/20 0.44
MAPK1 P28482 1/20 0.43
PNP P00491 1/20 0.43
TLR8 Q9NR97 4/20 0.41
DHFR P00374 1/20 0.40
ALDH1A1 P00352 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
HIF1A Q16665 1/20 0.40
PHLPP2 Q6ZVD8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7212493 0.88 ADORA2A (0.47) ADORA2AADORA1TLR7MAPK1PNP
SCHEMBL2060321 0.87 ADORA2A (0.46) ADORA2AADORA1TLR7MAPK1PNP
SCHEMBL14944613 0.87 ADORA2A (0.46) ADORA2AADORA1TLR7MAPK1PNP
SCHEMBL19370095 0.86 ADORA2A (0.45) ADORA2AADORA1TLR7MAPK1PNP
SCHEMBL5730944 0.86 TLR7 (0.55) ADORA2AADORA1TLR7MAPK1ALDH1A1
SCHEMBL5731043 0.85 ADORA1 (0.47) ADORA2AADORA1TLR7MAPK1PNP
SCHEMBL5731379 0.85 TLR7 (0.45) ADORA2AADORA1TLR7MAPK1PNP
SCHEMBL5731620 0.85 ADORA2A (0.59) ADORA2AADORA1TLR7MAPK1
SCHEMBL2060517 0.85 TLR7 (0.45) ADORA2AADORA1TLR7MAPK1PNP
SCHEMBL7209948 0.83 TSHR (0.52) ADORA2AADORA1TLR7MAPK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1035123-B1 NOVEL HETEROCYCLIC COMPOUNDS SUMITOMO PHARMA (JP) 2003-08-20 EP disclosed
US-6329381-B1 INTERFERONS, VIRICIDES AND ANTICARCINOGENIC AGENTS SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 2001-12-11 US disclosed
EP-1035123-A1 NOVEL HETEROCYCLIC COMPOUNDS SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 2000-09-13 EP disclosed