SCHEMBL7204863

SCHEMBL7204863

CCCCCN(C)CCCCCCO[C@H]1CC[C@H](N(C)S(=O)(=O)c2ccc([N+](=O)[O-])cc2)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.47
HTR2C P28335 3/20 0.47
LSS P48449 6/20 0.44
KCNH2 Q12809 3/20 0.42
CYP19A1 P11511 4/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPK1 P28482 1/20 0.41
KMT2A Q03164 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
MAPT P10636 1/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA3 P07451 1/20 0.38
CA4 P22748 1/20 0.38
CA6 P23280 1/20 0.38
CA5A P35218 1/20 0.38
CA7 P43166 1/20 0.38
CA9 Q16790 1/20 0.38
CA13 Q8N1Q1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7204860 1.00 HTR2A (0.47) HTR2AHTR2CLSSKCNH2CYP19A1
SCHEMBL7207309 0.99 HTR2A (0.47) HTR2AHTR2CLSSKCNH2CYP19A1
SCHEMBL7209122 0.99 HTR2A (0.47) HTR2AHTR2CLSSKCNH2CYP19A1
SCHEMBL4806400 0.89 CA12 (0.41) HTR2AHTR2CLSSKCNH2ALDH1A1
SCHEMBL4806405 0.89 CA12 (0.41) HTR2AHTR2CLSSKCNH2ALDH1A1
SCHEMBL4806143 0.88 LSS (0.56) HTR2AHTR2CLSSKCNH2ALDH1A1
SCHEMBL4806137 0.88 LSS (0.56) HTR2AHTR2CLSSKCNH2ALDH1A1
SCHEMBL7210657 0.87 HTR2A (0.49) HTR2AHTR2CLSSALDH1A1KMT2A
SCHEMBL7210651 0.87 HTR2A (0.49) HTR2AHTR2CLSSALDH1A1KMT2A
SCHEMBL7209344 0.87 HTR2A (0.50) HTR2AHTR2CLSSALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1311475-A1 NOVEL AMINOCYCLOHEXANE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2003-05-21 EP disclosed
WO-2002014267-A1 NOVEL AMINOCYCLOHEXANE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-02-21 WO disclosed