SCHEMBL7205095

SCHEMBL7205095

CCC(CC)Nc1nc(Cl)nc2c1ncn2[C@@H]1O[C@H](c2nc(C3CC3)no2)[C@H]2OC(C)(C)O[C@H]21

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 14/20 0.46
ADORA2A P29274 13/20 0.46
ADORA3 P0DMS8 10/20 0.46
HTR2C P28335 4/20 0.44
TMIGD3 P0DMS9 3/20 0.44
HTR2B P41595 3/20 0.44
ADORA2B P29275 4/20 0.41
HRH2 P25021 1/20 0.41
HTR5A P47898 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7206711 0.89 ADORA1 (0.46) ADORA1ADORA2AADORA3HTR2CTMIGD3
SCHEMBL7205475 0.88 ADORA1 (0.45) ADORA1ADORA2AADORA3HTR2CTMIGD3
SCHEMBL7099549 0.87 ADORA1 (0.47) ADORA1ADORA2AADORA3HTR2CTMIGD3
SCHEMBL6796905 0.86 ADORA1 (0.56) ADORA1ADORA2AADORA3HTR2CTMIGD3
Formic Acid SCHEMBL6574863 0.83 ADORA1 (0.52) ADORA1ADORA2AADORA3HTR2CTMIGD3
SCHEMBL6574869 0.81 ADORA1 (0.47) ADORA1ADORA2AADORA3HTR2CTMIGD3
SCHEMBL6574865 0.81 ADORA1 (0.47) ADORA1ADORA2AADORA3HTR2CTMIGD3
SCHEMBL6576609 0.79 PI4KA (0.43) ADORA1ADORA2AADORA3ADORA2B
SCHEMBL6839871 0.78 PI4KA (0.55) ADORA1ADORA2AADORA3HTR2CTMIGD3
SCHEMBL6839866 0.78 PI4KA (0.55) ADORA1ADORA2AADORA3HTR2CTMIGD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6610665-B1 Treatment of inflammatory diseases, asthma or chronic obstructive pulmonary disease SMITHKLINE BEECHAM CORPORATION 2003-08-26 US disclosed
EP-1056759-B1 2-(PURIN-9-YL) -TETRAHYDROFURAN-3, 4-DIOL DERIVATIVES GLAXO GROUP LTD (GB) 2002-09-04 EP disclosed