SCHEMBL7206263

SCHEMBL7206263

COc1cc2c(=O)[nH]cnc2cc1OCc1ccncc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 2/20 0.50
ERBB2 P04626 1/20 0.50
EPHA2 P29317 1/20 0.50
IP6K1 Q92551 2/20 0.48
FLT1 P17948 1/20 0.48
PDE10A Q9Y233 1/20 0.47
SRC P12931 1/20 0.47
CHEK1 O14757 3/20 0.43
KDM4A O75164 1/20 0.43
KDM4B O94953 1/20 0.43
KDM5C P41229 1/20 0.43
KDM4C Q9H3R0 1/20 0.43
KDM5B Q9UGL1 1/20 0.43
KDM3A Q9Y4C1 1/20 0.43
PDPK1 O15530 1/20 0.42
PLK1 P53350 1/20 0.42
ELANE P08246 1/20 0.42
CTSV O60911 1/20 0.42
CTSL P07711 1/20 0.42
KDM1A O60341 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL156504 0.89 IP6K1 (0.62) KDRIP6K1SRCPDPK1ELANE
SCHEMBL1013586 0.89 IP6K1 (0.62) KDRIP6K1SRCPDPK1ELANE
Hydrochloric Acid SCHEMBL27988350 0.88 IP6K1 (0.60) KDRIP6K1SRCPDPK1ELANE
SCHEMBL7460730 0.86 SRC (0.44) KDRERBB2EPHA2IP6K1FLT1
SCHEMBL5493946 0.84 SRC (0.46) KDRIP6K1PDE10ASRCCHEK1
SCHEMBL8917 0.83 SRC (0.63) IP6K1SRCCHEK1PDPK1PARP1
SCHEMBL20897397 0.82 IP6K1 (0.69) IP6K1CHEK1PDPK1ELANECTSV
SCHEMBL1781759 0.81 IP6K1 (0.58) KDRIP6K1PDPK1ELANECTSV
SCHEMBL1012421 0.80 SRC (0.55) IP6K1SRCCHEK1PARP1PIM1
SCHEMBL1014333 0.80 SRC (0.55) IP6K1SRCCHEK1PARP1PIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0912557-B1 OXINDOLE DERIVATIVES ASTRAZENECA AB (SE) 2003-07-09 EP disclosed
US-6362336-B1 ADMINISTERING A QUINAZOLINE DERIVATIVE TO A WARM-BLOODED ANIMAL FOR PRODUCING AN ANTIANGIOGENIC AND/OR VASCULAR PERMEABILITY REDUCING EFFECT ZENECA LIMITED (GB) 2002-03-26 US disclosed
US-20020032208-A1 Chemical compounds ZENECA LIMITED 2002-03-14 US disclosed
EP-0873319-B1 QUINAZOLINE DERIVATIVES ASTRAZENECA AB (SE) 2001-07-25 EP disclosed
US-6265411-B1 ANGIOGENESIS INHIBITOR ZENECA LIMITED (GB) 2001-07-24 US disclosed
US-6258951-B1 ANTICANCER, ANTIARTHRITIC AGENTS ZENECA LIMITED (GB) 2001-07-10 US disclosed
US-6071921-A Chemical compounds ZENECA LIMITED (GB) 2000-06-06 US disclosed
US-5962458-A ANGIOGENESIS INHIBITORS, ANTICANCER AGENTS, ANTIDIABETIC AGENTS, SKIN DISORDERS, AUTOIMMUNE DISEASES, ANTIINFLAMMATORY AGENTS, VISION DEFECTS ZENECA LIMITED (GB) 1999-10-05 US disclosed
EP-0912557-A1 OXINDOLE DERIVATIVES ZENECA LIMITED (GB) 1999-05-06 EP disclosed
EP-0873319-A1 QUINAZOLINE DERIVATIVES ZENECA LIMITED (GB) 1998-10-28 EP disclosed
WO-1997042187-A1 OXINDOLE DERIVATIVES ZENECA LIMITED (GB) 1997-11-13 WO disclosed
WO-1997022596-A1 QUINAZOLINE DERIVATIVES ZENECA LIMITED (GB) 1997-06-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020032208-A1 Chemical compounds FLT1, CNKSR1, KDR KDR 3/4885ERBB2 154/4885EPHA2 1014/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.