SCHEMBL7209433

SCHEMBL7209433

Nc1nc(SCc2ccccc2)nc2c1ncn2Cc1ccccc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.66
CYP1A2 P05177 1/20 0.66
CYP3A4 P08684 1/20 0.66
CYP2C9 P11712 1/20 0.66
CYP2C19 P33261 1/20 0.66
HIF1A Q16665 1/20 0.66
PHLPP2 Q6ZVD8 1/20 0.66
PDE4A P27815 1/20 0.60
PDE4B Q07343 1/20 0.60
PDE4C Q08493 1/20 0.60
PDE4D Q08499 1/20 0.60
ADORA2A P29274 3/20 0.58
PI4KA P42356 1/20 0.58
PI4K2B Q8TCG2 1/20 0.58
PI4K2A Q9BTU6 1/20 0.58
PI4KB Q9UBF8 1/20 0.58
ADORA3 P0DMS8 1/20 0.54
PNP P00491 1/20 0.52
NPC1 O15118 2/20 0.48
RAB9A P51151 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7211053 0.89 PDE4A (0.59) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL7212587 0.89 PDE4A (0.59) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL1286226 0.89 ADORA2A (0.58) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL7205568 0.88 PDE4A (0.58) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL7209300 0.86 PDE4A (0.57) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL7209247 0.86 PDE4A (0.62) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL7205020 0.86 PDE4A (0.62) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL7207338 0.85 PDE4A (0.56) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL7206475 0.85 PDE4D (0.56) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL7208530 0.84 PDE4A (0.55) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1035123-B1 NOVEL HETEROCYCLIC COMPOUNDS SUMITOMO PHARMA (JP) 2003-08-20 EP disclosed
US-6329381-B1 INTERFERONS, VIRICIDES AND ANTICARCINOGENIC AGENTS SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 2001-12-11 US disclosed
EP-1035123-A1 NOVEL HETEROCYCLIC COMPOUNDS SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 2000-09-13 EP disclosed