SCHEMBL7210973

SCHEMBL7210973

COc1ccc(N)cn1.Nc1cc[nH]n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.45
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
ALDH1A1 P00352 1/20 0.45
BRCA1 P38398 1/20 0.45
HBB P68871 1/20 0.45
HSD17B10 Q99714 1/20 0.45
NNMT P40261 1/20 0.40
POLB P06746 2/20 0.40
RAB9A P51151 1/20 0.40
KEAP1 Q14145 1/20 0.39
MKNK1 Q9BUB5 1/20 0.36
MKNK2 Q9HBH9 1/20 0.36
CYP2A6 P11509 1/20 0.35
PIK3CA P42336 3/20 0.35
PIK3CD O00329 2/20 0.35
PIK3CB P42338 2/20 0.35
PIK3CG P48736 2/20 0.35
PIP5K1C O60331 1/20 0.35
PI4KA P42356 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29536663 0.84
SCHEMBL113293 0.84
Hydrochloric Acid SCHEMBL5645807 0.82 KDM4E (0.56) KDM4EMEN1KMT2AALDH1A1BRCA1
Hydrochloric Acid SCHEMBL5649941 0.82 KDM4E (0.56) KDM4EMEN1KMT2AALDH1A1BRCA1
Formaldehyde SCHEMBL28810279 0.78 KDM4E (0.53) KDM4EMEN1KMT2AALDH1A1BRCA1
SCHEMBL28238027 0.73
SCHEMBL956 0.73
Methyl Alcohol SCHEMBL28819104 0.71
SCHEMBL16835945 0.71 MKNK1 (0.51) KDM4EMEN1KMT2AALDH1A1BRCA1
Hydrochloric Acid SCHEMBL3832185 0.71

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1339702-A1 5-AMIDE SUBSTITUTED DIARYLAMINES AS MEK INHIBITORS WARNER-LAMBERT COMPANY (US) 2003-09-03 EP disclosed
WO-2001068619-A1 5-AMIDE SUBSTITUTED DIARYLAMINES AS MEX INHIBITORS WARNER-LAMBERT COMPANY (US) 2001-09-20 WO disclosed