SCHEMBL7216505

SCHEMBL7216505

COC(=O)C1=Cc2cc(OCc3ccc(Cl)cc3)ccc2S(=O)(=O)CC1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
MAOB P27338 7/20 0.43
MAOA P21397 6/20 0.43
KDM5A P29375 1/20 0.40
KDM5B Q9UGL1 1/20 0.40
NR4A2 P43354 2/20 0.39
KMT2A Q03164 2/20 0.39
MEN1 O00255 1/20 0.39
HSP90AA1 P07900 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
HTT P42858 1/20 0.39
PPARD Q03181 1/20 0.38
PPARA Q07869 1/20 0.38
SLC26A4 O43511 1/20 0.38
SMPD1 P17405 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7222605 0.91 MAOB (0.44) MAOBMAOAKDM5AKDM5BNR4A2
SCHEMBL7218066 0.90 NPC1 (0.41) NPC1RAB9AKMT2AMEN1HSP90AA1
SCHEMBL7218316 0.89 NR4A2 (0.47) NPC1RAB9AMAOBMAOANR4A2
SCHEMBL7218242 0.87 NPC1 (0.37) NPC1RAB9AKMT2AMEN1HSP90AA1
SCHEMBL7222803 0.85 NPC1 (0.38) NPC1RAB9AKMT2AMEN1HSP90AA1
SCHEMBL7215817 0.85 NPC1 (0.38) NPC1RAB9AKMT2AMEN1HSP90AA1
SCHEMBL7222229 0.84 S1PR1 (0.40) NPC1RAB9AKMT2AMEN1MAPT
SCHEMBL7216612 0.84 MAOB (0.43) NPC1RAB9AMAOBMAOANR4A2
SCHEMBL7222460 0.84 MRGPRX4 (0.47) NPC1RAB9AMAOB
SCHEMBL7222083 0.83 MRGPRX4 (0.46) NPC1RAB9AMAOBMAOAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6627651-B1 Exhibiting preventive and therapeutic effects against HIV infectious diseases wherein R1 is an optionally substituted five- or six-membered ring group; X1 is a free valency or the like; W is a divalent group and inhibitors of HIV (human TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-09-30 US disclosed
EP-1182195-A1 CYCLIC COMPOUNDS AND USES THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-02-27 EP disclosed