SCHEMBL7217024

SCHEMBL7217024

O=C(Nc1ccn(CCCNC2CCC2)n1)c1c[nH]c2c1-c1ncccc1CCC2

nearest known ligand 0.31

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 1/20 0.31
PDE4D Q08499 1/20 0.31
GCK P35557 1/20 0.31
NPSR1 Q6W5P4 1/20 0.30
GRIN1 Q05586 1/20 0.30
GRIN2B Q13224 1/20 0.30
IDO1 P14902 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7223193 0.89 PIM1 (0.32) PDE4BPDE4DGCKNPSR1
SCHEMBL7218337 0.88 GCK (0.33) PDE4BPDE4DGCKNPSR1
SCHEMBL7223026 0.88 GCK (0.33) PDE4BPDE4DGCKNPSR1
SCHEMBL7223477 0.87 HRH4 (0.30)
SCHEMBL7221707 0.87 GCK (0.32) GCKNPSR1
SCHEMBL7223214 0.86 NPSR1 (0.34) PDE4BPDE4DGCKNPSR1
SCHEMBL7216130 0.86 GCK (0.36) GCKNPSR1
SCHEMBL7222958 0.86 NPSR1 (0.34) PDE4BPDE4DGCKNPSR1
SCHEMBL7222537 0.85 GCK (0.32) GCKNPSR1
SCHEMBL7222707 0.85 GCK (0.34) PDE4BPDE4DGCKNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6653471-B2 Tricyclic heteroaromatic compounds containing pyrrole ring; central nervous system disorder treatment; side effect reduction NEUROGEN CORPORATION 2003-11-25 US disclosed