SCHEMBL7217112

SCHEMBL7217112

CCOc1ccc2nc(N)sc2c1.Cc1cc(N)no1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 7/20 0.74
TP53 P04637 4/20 0.74
HSD17B10 Q99714 3/20 0.74
TSHR P16473 2/20 0.74
ALDH1A1 P00352 2/20 0.74
KMT2A Q03164 3/20 0.55
CYP1A2 P05177 3/20 0.52
CYP2C19 P33261 2/20 0.52
RAB9A P51151 7/20 0.51
NPC1 O15118 6/20 0.51
LMNA P02545 4/20 0.50
PKM P14618 2/20 0.50
KDM4E B2RXH2 1/20 0.50
CA12 O43570 1/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
CA3 P07451 1/20 0.50
CA4 P22748 1/20 0.50
CA6 P23280 1/20 0.50
CA5A P35218 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL233589 0.86 CYP3A4 (1.00) CYP3A4TP53HSD17B10TSHRALDH1A1
SCHEMBL8129225 0.79 CYP3A4 (0.84) CYP3A4TP53HSD17B10TSHRALDH1A1
SCHEMBL9722752 0.75 CYP3A4 (0.78) CYP3A4TP53HSD17B10TSHRALDH1A1
SCHEMBL5946843 0.75 CYP3A4 (0.78) CYP3A4TP53HSD17B10TSHRALDH1A1
SCHEMBL31257148 0.75 CYP3A4 (0.77) CYP3A4TP53HSD17B10TSHRALDH1A1
SCHEMBL482497 0.75 CYP3A4 (0.77) CYP3A4TP53HSD17B10TSHRALDH1A1
Hydrochloric Acid SCHEMBL11613963 0.74 CYP3A4 (0.76) CYP3A4TP53HSD17B10TSHRALDH1A1
SCHEMBL8261943 0.73 KMT2A (0.69) CYP3A4TP53HSD17B10TSHRALDH1A1
SCHEMBL1748243 0.72 KMT2A (1.00) CYP3A4TP53HSD17B10TSHRALDH1A1
SCHEMBL11344342 0.72 CYP3A4 (0.72) CYP3A4TP53HSD17B10TSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1339702-A1 5-AMIDE SUBSTITUTED DIARYLAMINES AS MEK INHIBITORS WARNER-LAMBERT COMPANY (US) 2003-09-03 EP disclosed
WO-2001068619-A1 5-AMIDE SUBSTITUTED DIARYLAMINES AS MEX INHIBITORS WARNER-LAMBERT COMPANY (US) 2001-09-20 WO disclosed