SCHEMBL7217432

SCHEMBL7217432

CCCCCCC=C(Oc1ccccc1)C(=O)O

nearest known ligand 0.50

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ZDHHC2 Q9UIJ5 1/20 0.50
EP300 Q09472 1/20 0.49
FAAH O00519 7/20 0.46
PPARA Q07869 3/20 0.43
SOAT2 O75908 1/20 0.43
SOAT1 P35610 1/20 0.43
PPARG P37231 2/20 0.42
EPHX2 P34913 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22323840 1.00 ZDHHC2 (0.50) ZDHHC2EP300FAAHPPARASOAT2
SCHEMBL9781746 1.00 ZDHHC2 (0.50) ZDHHC2EP300FAAHPPARASOAT2
SCHEMBL22323843 1.00 ZDHHC2 (0.50) ZDHHC2EP300FAAHPPARASOAT2
SCHEMBL22323842 1.00 ZDHHC2 (0.50) ZDHHC2EP300FAAHPPARASOAT2
SCHEMBL22323852 0.98 ZDHHC2 (0.48) ZDHHC2EP300FAAHPPARASOAT2
SCHEMBL22323853 0.98 ZDHHC2 (0.48) ZDHHC2EP300FAAHPPARASOAT2
SCHEMBL22323850 0.87 ZDHHC2 (0.41) ZDHHC2FAAH
SCHEMBL22323848 0.87 ZDHHC2 (0.41) ZDHHC2FAAH
SCHEMBL4218119 0.87 ZDHHC2 (0.41) ZDHHC2FAAH
SCHEMBL2831627 0.86 ZDHHC2 (0.46) ZDHHC2EP300FAAHPPARASOAT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177227-B1 WATER PLASTICIZED HIGH REFRACTIVE INDEX POLYMER FOR OPHTHALMIC APPLICATIONS SURGIDEV CORP (US) 2003-10-01 EP claimed
US-11931365-B2 Use of PPAR-delta agonists in the treatment of disease RENEO PHARMACEUTICALS, INC. (US) 2024-03-19 US disclosed
US-20240016809-A1 USE OF PPAR-DELTA AGONISTS IN THE TREATMENT OF DISEASE RENEO PHARMACEUTICALS, INC. 2024-01-18 US disclosed
WO-2023147309-A1 USE OF PPAR-DELTA AGONISTS IN THE TREATMENT OF DISEASE RENEO PHARMACEUTICALS, INC. (US) 2023-08-03 WO disclosed
US-20230233570-A1 USE OF PPAR-DELTA AGONISTS IN THE TREATMENT OF DISEASE RENEO PHARMACEUTICALS, INC. 2023-07-27 US disclosed
US-20220370467-A1 USING OF A PPAR-DELTA AGONIST IN THE TREATMENT OF KIDNEY DISEASE WASHINGTON UNIVERSITY 2022-11-24 US disclosed
EP-4031124-A1 USE OF A PPAR-DELTA AGONIST IN THE TREATMENT OF KIDNEY DISEASE Reneo Pharmaceuticals, Inc. (US) 2022-07-27 EP disclosed
CN-114727976-A Use of PPAR-delta agonists in the treatment of renal disease 雷内奥制药公司 2022-07-08 CN disclosed
US-20220117972-A1 USE OF PPAR-DELTA AGONISTS IN THE TREATMENT OF MITOCHONDRIAL MYOPATHY RENEO PHARMACEUTICALS, INC. 2022-04-21 US disclosed
US-20220023306-A1 USE OF A PPAR-DELTA AGONIST IN THE TREATMENT OF FATTY ACID OXIDATION DISORDERS (FAOD) RENEO PHARMACEUTICALS, INC. 2022-01-27 US disclosed
EP-3927718-A1 USE OF PPAR-DELTA AGONISTS IN THE TREATMENT OF MITOCHONDRIAL MYOPATHY Reneo Pharmaceuticals, Inc. (US) 2021-12-29 EP disclosed
EP-3920903-A1 USE OF A PPAR-DELTA AGONIST IN THE TREATMENT OF FATTY ACID OXIDATION DISORDERS (FAOD) Reneo Pharmaceuticals, Inc. (US) 2021-12-15 EP disclosed
CN-113747891-A Use of PPAR delta agonists in the treatment of Fatty Acid Oxidation Disorders (FAOD) 雷内奥制药公司 2021-12-03 CN disclosed
CN-113710683-A Use of PPAR-delta agonists in the treatment of mitochondrial myopathy 雷内奥制药公司 2021-11-26 CN disclosed
WO-2021055725-A1 USE OF A PPAR-DELTA AGONIST IN THE TREATMENT OF KIDNEY DISEASE RENEO PHARMACEUTICALS, INC. (US) 2021-03-25 WO disclosed
WO-2020163240-A1 USE OF A PPAR-DELTA AGONIST IN THE TREATMENT OF FATTY ACID OXIDATION DISORDERS (FAOD) RENEO PHARMACEUTICALS, INC. (US) 2020-08-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220370467-A1 USING OF A PPAR-DELTA AGONIST IN THE TREATMENT OF KIDNEY DISEASE PPARG, PPARA, PPARD ZDHHC2 749/4885EP300 247/4885FAAH 416/4885
US-11931365-B2 Use of PPAR-delta agonists in the treatment of disease PPARG, PPARD, PPARA ZDHHC2 434/4885EP300 152/4885FAAH 748/4885
US-20230233570-A1 USE OF PPAR-DELTA AGONISTS IN THE TREATMENT OF DISEASE PPARG, PPARD, PPARA ZDHHC2 434/4885EP300 152/4885FAAH 748/4885
US-20220117972-A1 USE OF PPAR-DELTA AGONISTS IN THE TREATMENT OF MITOCHONDRIAL MYOPATHY PPARD, PPARA, MTPN ZDHHC2 831/4885EP300 1686/4885FAAH 1062/4885
US-20240016809-A1 USE OF PPAR-DELTA AGONISTS IN THE TREATMENT OF DISEASE PPARG, PPARD, PPARA ZDHHC2 434/4885EP300 152/4885FAAH 748/4885
US-20220023306-A1 USE OF A PPAR-DELTA AGONIST IN THE TREATMENT OF FATTY ACID OXIDATION DISORDERS (FAOD) PPARD, ACOX1, CPT1A ZDHHC2 212/4885EP300 936/4885FAAH 354/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.