SCHEMBL7217488

SCHEMBL7217488

Oc1ccc2[nH]c(C3CCNCC3)nc2c1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 5/20 0.46
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
KDM4E B2RXH2 1/20 0.40
MAPT P10636 1/20 0.40
GFER P55789 1/20 0.40
USP7 Q93009 4/20 0.40
QDPR P09417 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CHEK1 O14757 1/20 0.37
WEE1 P30291 1/20 0.37
TLR9 Q9NR96 1/20 0.36
TLR8 Q9NR97 1/20 0.36
TLR7 Q9NYK1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7968684 0.82 PARP1 (0.43) PARP1NPC1RAB9AKDM4EMAPT
SCHEMBL2589997 0.82 CDC7 (0.48) PARP1NPC1RAB9AKDM4EMAPT
SCHEMBL3728479 0.82 PARP1 (0.43) PARP1NPC1RAB9AKDM4EMAPT
SCHEMBL2595517 0.82 TLR9 (0.48) PARP1NPC1RAB9AQDPRTLR9
SCHEMBL2111216 0.82 NPC1 (0.58) PARP1NPC1RAB9AKDM4EMAPT
SCHEMBL1298735 0.82 PARP1 (0.49) PARP1NPC1RAB9AKDM4EMAPT
SCHEMBL14447538 0.82 NPC1 (0.51) PARP1NPC1RAB9AKDM4EMAPT
SCHEMBL14447528 0.82 KDM4E (0.57) PARP1NPC1RAB9AKDM4EMAPT
Hydrochloric Acid SCHEMBL1981017 0.81 CDC7 (0.47) PARP1NPC1RAB9AKDM4EMAPT
Hydrochloric Acid SCHEMBL1299402 0.81 PARP1 (0.48) PARP1NPC1RAB9AKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6660751-B1 Sulfonamide derivatives as 5-HT7 receptor antagonists SMITHKLINE BEECHAM P.L.C. (GB) 2003-12-09 US disclosed