SCHEMBL7218612

SCHEMBL7218612

COc1cc2c(cc1OC)C(Cc1ccc3ccccc3c1)N(CC(=O)N1CCc3ccccc3C1)CC2

nearest known ligand 0.86

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 20/20 0.86
HCRTR2 O43614 16/20 0.86

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6786780 0.82 HCRTR1 (0.87) HCRTR1HCRTR2
SCHEMBL6376207 0.81 HCRTR1 (0.86) HCRTR1HCRTR2
SCHEMBL6375492 0.80 HCRTR1 (0.87) HCRTR1HCRTR2
SCHEMBL6787039 0.80 HCRTR1 (0.87) HCRTR1HCRTR2
SCHEMBL6374586 0.79 HCRTR1 (0.72) HCRTR1HCRTR2
SCHEMBL6790070 0.78 HCRTR1 (0.67) HCRTR1HCRTR2
SCHEMBL6789272 0.78 HCRTR1 (0.67) HCRTR1HCRTR2
SCHEMBL6376319 0.77 HCRTR1 (0.72) HCRTR1HCRTR2
SCHEMBL6382603 0.77 HCRTR1 (0.88) HCRTR1HCRTR2
SCHEMBL6375236 0.76 HCRTR1 (0.67) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1274687-A1 1,2,3,4- TETRAHYDROISOQUINOLINE DERIVATIVES Actelion Pharmaceuticals Ltd. (CH) 2003-01-15 EP disclosed
WO-2001068609-A1 1,2,3,4-TETRAHYDROISOQUINOLINE DERIVATIVES ACTELION PHARMACEUTICALS LTD. (CH) 2001-09-20 WO disclosed