SCHEMBL7219759

SCHEMBL7219759

CC(C)c1cc2nc(C(=O)O)nn2nc1OCCCN1CCC(OC(c2ccccc2)c2ccccc2)CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 10/20 0.51
PARP14 Q460N5 2/20 0.48
CHRM2 P08172 2/20 0.45
HTR1A P08908 2/20 0.45
ADRA2A P08913 2/20 0.45
CHRM1 P11229 2/20 0.45
DRD1 P21728 2/20 0.45
SLC6A2 P23975 2/20 0.45
ADRA1A P35348 2/20 0.45
DRD3 P35462 2/20 0.45
SLC6A3 Q01959 2/20 0.45
KCNH2 Q12809 2/20 0.45
NPC1 O15118 1/20 0.45
MLNR O43193 1/20 0.45
NR1I2 O75469 1/20 0.45
EGFR P00533 1/20 0.45
LMNA P02545 1/20 0.45
ERBB2 P04626 1/20 0.45
FYN P06241 1/20 0.45
CHRM4 P08173 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6621233 0.84 PARP14 (0.51) BCHEPARP14CHRM2HTR1AADRA2A
Fumaric Acid SCHEMBL7009266 0.84 BCHE (0.50) BCHEPARP14CHRM2HTR1AADRA2A
Fumaric Acid SCHEMBL7227367 0.84 BCHE (0.50) BCHEPARP14CHRM2HTR1AADRA2A
SCHEMBL6619355 0.84 PARP14 (0.63) BCHEPARP14CHRM2HTR1AADRA2A
SCHEMBL7219755 0.78 PARP14 (0.59) BCHEPARP14CHRM2HTR1AADRA2A
SCHEMBL7218894 0.78 CHRM2 (0.49) BCHEPARP14CHRM2HTR1AADRA2A
SCHEMBL6619594 0.77 PARP14 (0.61) BCHEPARP14CHRM2HTR1AADRA2A
SCHEMBL6621846 0.73 PARP14 (0.48) BCHEPARP14CHRM2HTR1AADRA2A
Hydrochloric Acid SCHEMBL6618531 0.72 BCHE (0.51) BCHEPARP14CHRM2HTR1AADRA2A
SCHEMBL6621948 0.72 PARP14 (0.58) BCHEPARP14CHRM2HTR1AADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6627630-B1 Preventing or treating allergic skin diseases such as contact dermatitis, pruritus, dried dermatitis, acute urticaria prurigo and antiallergins TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-09-30 US disclosed