SCHEMBL7220901

SCHEMBL7220901

CC1(c2ccc(O)cc2)COc2cc(O)ccc2C1CCCCCCCCCC(CCCC(F)(F)C(F)(F)C(F)(F)C(F)(F)F)C(=O)O

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.54
AR P10275 1/20 0.33
TMEM97 Q5BJF2 2/20 0.31
NR1I2 O75469 1/20 0.30
NR3C1 P04150 1/20 0.30
PGR P06401 1/20 0.30
ESRRA P11474 1/20 0.30
EPHX2 P34913 1/20 0.30
PPARG P37231 1/20 0.30
ESR2 Q92731 1/20 0.30
NR1H4 Q96RI1 1/20 0.30
SIRT5 Q9NXA8 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
ALOX15 P16050 1/20 0.30
CYP2C19 P33261 1/20 0.30
HTR2B P41595 1/20 0.30
SIGMAR1 Q99720 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7224589 1.00 ESR1 (0.54) ESR1ARTMEM97NR1I2NR3C1
SCHEMBL7218943 0.98 ESR1 (0.52) ESR1ARTMEM97
SCHEMBL7220866 0.98 ESR1 (0.52) ESR1ARTMEM97
SCHEMBL5854406 0.94 ESR1 (0.47) ESR1ARTMEM97NR1I2NR3C1
SCHEMBL5855481 0.94 ESR1 (0.47) ESR1ARTMEM97NR1I2NR3C1
SCHEMBL5856044 0.94 ESR1 (0.47) ESR1ARTMEM97NR1I2NR3C1
SCHEMBL5854247 0.94 ESR1 (0.47) ESR1ARTMEM97NR1I2NR3C1
SCHEMBL5854200 0.94 ESR1 (0.47) ESR1ARTMEM97NR1I2NR3C1
SCHEMBL5854630 0.94 ESR1 (0.47) ESR1ARTMEM97NR1I2NR3C1
SCHEMBL5853959 0.94 ESR1 (0.47) ESR1ARTMEM97NR1I2NR3C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6552069-B1 Having anti-estrogenic activity; for use in therapy CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-04-22 US claimed
EP-1241166-A1 3-METHYL-CHROMAN AND -THIOCHROMAN DERIVATIVES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2002-09-18 EP claimed
US-6552069-B1 Having anti-estrogenic activity; for use in therapy CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-04-22 US disclosed
EP-1241166-A1 3-METHYL-CHROMAN AND -THIOCHROMAN DERIVATIVES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2002-09-18 EP disclosed