SCHEMBL7220947

SCHEMBL7220947

CN(C)CCC#CC(=O)Nc1ccc2ncnc(Nc3cccc(Br)c3)c2c1

nearest known ligand 0.83

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
EGFR P00533 20/20 0.83
ERBB2 P04626 18/20 0.83
ERBB4 Q15303 2/20 0.75
ABCG2 Q9UNQ0 1/20 0.75

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7220938 0.96 EGFR (0.81) EGFRERBB2ERBB4ABCG2
SCHEMBL7214783 0.96 EGFR (0.79) EGFRERBB2ERBB4ABCG2
SCHEMBL30115365 0.91 EGFR (1.00) EGFRERBB2ERBB4ABCG2
SCHEMBL7214823 0.89 EGFR (0.68) EGFRERBB2ERBB4
SCHEMBL30115314 0.87 EGFR (1.00) EGFRERBB2ERBB4ABCG2
SCHEMBL30115332 0.86 EGFR (0.84) EGFRERBB2ERBB4ABCG2
SCHEMBL29350449 0.86 EGFR (1.00) EGFRERBB2ERBB4ABCG2
SCHEMBL29350915 0.86 EGFR (1.00) EGFRERBB2ERBB4ABCG2
SCHEMBL412104 0.86 EGFR (1.00) EGFRERBB2ERBB4ABCG2
SCHEMBL7782260 0.86 EGFR (1.00) EGFRERBB2ERBB4ABCG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6602863-B1 Irreversible inhibitors of tyrosine kinases WARNER-LAMBERT COMPANY 2003-08-05 US disclosed